FAIRMol

Reverse docking explorer

Search one compound across many targets or scan the strongest compound-target pairs in the active database. The combined reverse-docking score uses a normalized docking-score estimator together with an interaction-fingerprint component.

DB SELECTIONExplorer results are being read from this database.
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1 compounds in matrix 15 best compound-target hits listed 15 targets
• Combined reverse-docking score = 65% normalized docking-score estimator + 35% interaction-fingerprint component.
• When a native ligand exists for an experiment, the interaction-fingerprint component is driven by similarity to the native contact/H-bond pattern.
• When no native ligand exists, the interaction-fingerprint component falls back to contact richness within the experiment (normalized contacts and H-bonds).

Compounds × targets matrix

Each cell shows the best combined reverse-docking score found for that compound on that target. Blank cells mean no imported pose passed the current filters.
Compound Best Mean Targets T03T05T09T11T12T13T14T15T16T17T18T19T20T21T22
GemmaOHDUnisi_41 0.883 0.809 15 0.79 0.83 0.76 0.88 0.88 0.77 0.79 0.80 0.82 0.78 0.82 0.72 0.78 0.86 0.86

Best compound-target hits

The score column is the combined reverse-docking score. The next two columns expose its components: normalized score-estimator and interaction fingerprint.
CompoundTargetExperimentCombinedScore partIFP partIFP modeMetricDock scoreInter normContactsHB
GemmaOHDUnisi_41 T12
native IFP available
T12
selection_import_t12
0.883 1.000 0.667 native_similarity final_rank_score -26.2423 -0.810312 20 7 Pose
GemmaOHDUnisi_41 T11
native IFP available
T11
selection_import_t11
0.877 1.000 0.649 native_similarity final_rank_score -24.1764 -0.695149 10 7 Pose
GemmaOHDUnisi_41 T21
native IFP available
T21
selection_import_t21
0.865 1.000 0.614 native_similarity final_rank_score -27.9819 -0.751309 17 5 Pose
GemmaOHDUnisi_41 T22
native IFP available
T22
selection_import_t22
0.861 1.000 0.604 native_similarity final_rank_score -33.7094 -0.940685 24 11 Pose
GemmaOHDUnisi_41 T05
native IFP available
T05
selection_import_t05
0.826 1.000 0.503 native_similarity final_rank_score -29.8668 -0.837854 13 7 Pose
GemmaOHDUnisi_41 T18
native IFP available
T18
selection_import_t18
0.820 1.000 0.485 native_similarity final_rank_score -15.5491 -0.595751 17 3 Pose
GemmaOHDUnisi_41 T16
native IFP available
T16
selection_import_t16
0.815 1.000 0.472 native_similarity final_rank_score -23.4933 -0.65678 16 3 Pose
GemmaOHDUnisi_41 T15
native IFP available
T15
selection_import_t15
0.797 1.000 0.421 native_similarity final_rank_score -25.2904 -0.836742 18 4 Pose
GemmaOHDUnisi_41 T03
native IFP available
T03
selection_import_t03
0.790 1.000 0.401 native_similarity final_rank_score -26.102 -0.841444 16 8 Pose
GemmaOHDUnisi_41 T14
native IFP available
T14
selection_import_t14
0.785 1.000 0.387 native_similarity final_rank_score -19.3542 -0.632747 19 9 Pose
GemmaOHDUnisi_41 T17
native IFP available
T17
selection_import_t17
0.781 1.000 0.375 native_similarity final_rank_score -29.818 -0.749818 21 7 Pose
GemmaOHDUnisi_41 T20
native IFP available
T20
selection_import_t20
0.778 1.000 0.366 native_similarity final_rank_score -22.5384 -0.60587 15 8 Pose
GemmaOHDUnisi_41 T13
native IFP available
T13
selection_import_t13
0.769 1.000 0.339 native_similarity final_rank_score -23.6613 -0.790161 20 11 Pose
GemmaOHDUnisi_41 T09
native IFP available
T09
selection_import_t09
0.762 1.000 0.320 native_similarity final_rank_score -29.6374 -0.819328 17 5 Pose
GemmaOHDUnisi_41 T19
native IFP available
T19
selection_import_t19
0.723 1.000 0.209 native_similarity final_rank_score -31.9318 -0.974129 22 5 Pose