FAIRMol

Z86240607

Pose ID 7966 Compound 767 Pose 1379

DB Docking_panel_21Docking pose analysis is being read from this database.
Molecular metrics status: done
Cached molecular metrics are available for this pose.
Metrics cached · SASA missing
T04
Pteridine reductase 1 (PTR1) Leishmania major
Ligand Z86240607
PDB7PXX

3D complex viewer

Strict H-bonds Permissive H-bonds
Viewer legend
Protein receptor
Pocket residues
Cofactor context
Docked ligand
Overall assessment
Weak No SASA yet
Weak or marginal quality
Binding strong Geometry high Native mixed SASA missing
Strain ΔE
10.2 kcal/mol
Protein clashes
1
Internal clashes
2
Native overlap
contact recall 0.53, Jaccard 0.53, H-bond role recall 0.20
Burial
92%
Reason: no major geometry red flags detected
1 protein-contact clashes
Molecular report
Full metrics ↗
Weak Marginal quality. Consider only alongside better-scoring alternatives.
✓ Excellent LE (-1.267 kcal/mol/HA) ✓ Good fit quality (FQ -10.15) ✗ Moderate strain (10.2 kcal/mol) ✗ Geometry warnings ✗ Protein-contact clashes (6) ℹ SASA not computed
Score
-22.802
kcal/mol
LE
-1.267
kcal/mol/HA
Fit Quality
-10.15
FQ (Leeson)
HAC
18
heavy atoms
MW
258
Da
LogP
3.00
cLogP
Strain ΔE
10.2 kcal/mol
SASA buried
computing…

Interaction summary

HB 2 HY 14 PI 3 CLASH 2
Final rank1.498Score-22.802
Inter norm-1.305Intra norm0.039
Top1000noExcludedno
Contacts10H-bonds1
Artifact reasongeometry warning; 3 clashes; 6 protein contact clashes
Residues
ARG17 HIS241 LEU188 LEU226 LEU229 NDP302 PHE113 TYR191 TYR194 ARG287

Protein summary

308 residues
Protein targetT04Atoms4210
Residues308Chains3
Residue summaryLEU:494; ALA:421; ARG:384; VAL:368; THR:295; TYR:231; SER:198; PRO:196; ILE:190; LYS:176; ASN:154; GLU:150; GLY:126; PHE:120; HIS:119; ASP:108

Receptor context

1 kept / 0 excluded
Receptor context filtering: interactions and SASA are computed against protein atoms plus allowed cofactors/ions. Native ligand-like HETATM partners are excluded from scoring.
Kept context 1 Excluded HETATM 0
Kept cofactors / ions
A:NDP302

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: permissive.
Name7PXXContacts19
PoseOpen native poseHB0
IFP residues
ARG17 ASP181 GLY225 HIS241 LEU188 LEU226 LEU229 LYS198 MET233 NDP302 PHE113 PRO115 SER111 SER112 SER227 TYR191 TYR194 VAL230 ARG287
Current overlap10Native recall0.53
Jaccard0.53RMSD-
HB strict1Strict recall0.17
HB same residue+role1HB role recall0.20
HB same residue1HB residue recall0.20

HB · H-bonds

Mode: permissive. Count shows atom-level H-bonds; unique residues in summary: 0.

PI · π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

HY · Hydrophobic contacts

CLASH · Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBCTCT overlapCT recallHB role rec.RMSDExcluded
1379 1.4983702612961016 -1.30538 -22.8022 1 10 10 0.53 0.20 - no Current

Molecular metrics

RDKit SASA burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -22.802kcal/mol
Ligand efficiency (LE) -1.2668kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -10.152
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 18HA

Physicochemical properties

Molecular weight 258.4Da
Lipinski: ≤ 500 Da
LogP (cLogP) 3.00
Lipinski: ≤ 5
Rotatable bonds 5

Conformational strain (MMFF94s)

Strain energy (ΔE) 10.16kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy -6.76kcal/mol
Minimised FF energy -16.92kcal/mol

SASA & burial

not yet run
SASA has not been computed yet for this pose. Queue a background recompute to populate SASA burial metrics without blocking the page.