FAIRMol

OSA_Lib_28

Pose ID 4118 Compound 84 Pose 800

DB Docking_panel_21Docking pose analysis is being read from this database.
Molecular metrics status: done
Cached molecular metrics are available for this pose.
Metrics cached · SASA missing
T03
Bifunctional dihydrofolate reductase-thymidylate synthase (DHFR-TS) 'ambiguous: archive label suggests Leishmania major, structure title points to Trypanosoma cruzi template'
Ligand OSA_Lib_28
PDB3CL9

3D complex viewer

Strict H-bonds Permissive H-bonds
Viewer legend
Protein receptor
Pocket residues
Cofactor context
Docked ligand
Overall assessment
Weak No SASA yet
Weak or marginal quality
Binding strong Geometry medium Native strong SASA missing
Strain ΔE
19.2 kcal/mol
Protein clashes
4
Internal clashes
4
Native overlap
contact recall 0.80, Jaccard 0.70, H-bond role recall 0.00
Burial
96%
Reason: no major geometry red flags detected
4 protein-contact clashes 4 intramolecular clashes
Molecular report
Full metrics ↗
Weak Marginal quality. Consider only alongside better-scoring alternatives.
✓ Excellent LE (-0.746 kcal/mol/HA) ✓ Good fit quality (FQ -7.33) ✗ Moderate strain (19.2 kcal/mol) ✗ Geometry warnings ✗ Many internal clashes (18) ✗ Excluded by docking heuristics ℹ SASA not computed
Score
-23.866
kcal/mol
LE
-0.746
kcal/mol/HA
Fit Quality
-7.33
FQ (Leeson)
HAC
32
heavy atoms
MW
423
Da
LogP
3.87
cLogP
Strain ΔE
19.2 kcal/mol
SASA buried
computing…

Interaction summary

HB 2 HY 24 PI 2 CLASH 4
Final rank6.829Score-23.866
Inter norm-0.797Intra norm0.052
Top1000noExcludedyes
Contacts19H-bonds0
Artifact reasonexcluded; geometry warning; 18 clashes; 1 protein clash; moderate strain Δ 19.3
Residues
ALA32 ARG48 ASP52 ILE45 LEU94 MET53 NDP301 PHE56 PRO88 SER86 THR180 THR83 TRP47 TYR162 VAL156 VAL30 VAL31 VAL49 VAL87

Protein summary

225 residues
Protein targetT03Atoms3428
Residues225Chains2
Residue summaryLEU:380; ARG:360; VAL:272; LYS:264; ALA:240; GLU:240; PRO:224; PHE:180; THR:154; ILE:152; SER:132; TYR:126; GLN:119; ASN:98; GLY:84; NDP:74

Receptor context

1 kept / 0 excluded
Receptor context filtering: interactions and SASA are computed against protein atoms plus allowed cofactors/ions. Native ligand-like HETATM partners are excluded from scoring.
Kept context 1 Excluded HETATM 0
Kept cofactors / ions
A:NDP301

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: permissive.
Name3CL9Contacts20
PoseOpen native poseHB0
IFP residues
ALA32 ARG97 ASP52 ILE45 LEU94 LYS57 MET53 NDP301 PHE56 PHE91 PRO88 SER86 THR180 THR54 THR83 TYR162 VAL156 VAL30 VAL31 VAL87
Current overlap16Native recall0.80
Jaccard0.70RMSD-
HB strict0Strict recall0.00
HB same residue+role0HB role recall0.00
HB same residue0HB residue recall0.00

HB · H-bonds

Mode: permissive. Count shows atom-level H-bonds; unique residues in summary: 0.

PI · π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

HY · Hydrophobic contacts

CLASH · Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBCTCT overlapCT recallHB role rec.RMSDExcluded
882 3.68015874069592 -0.758599 -23.1905 0 17 0 0.00 0.00 - no Open
618 4.753718222757358 -0.879782 -27.9333 0 11 0 0.00 0.00 - no Open
880 4.760586587214268 -0.789752 -25.2392 0 19 0 0.00 0.00 - no Open
876 4.865720514621524 -0.80982 -25.2682 0 19 0 0.00 0.00 - no Open
614 5.2705305231790405 -0.881861 -28.2029 0 11 0 0.00 0.00 - no Open
806 5.387341035556807 -0.80016 -25.685 0 18 15 0.75 0.00 - no Open
878 5.717936949193543 -0.823674 -25.1139 0 21 0 0.00 0.00 - no Open
610 5.896851545489233 -0.88753 -28.019 1 13 0 0.00 0.00 - no Open
609 5.912714715887796 -1.02151 -29.0331 1 18 0 0.00 0.00 - no Open
883 7.483230480035522 -0.74954 -21.634 0 19 0 0.00 0.00 - no Open
611 7.781050852582138 -1.01052 -24.7664 1 16 0 0.00 0.00 - no Open
613 8.164514631771638 -0.879609 -27.0241 0 17 0 0.00 0.00 - no Open
615 5.871673633146488 -1.02301 -27.44 0 15 0 0.00 0.00 - yes Open
801 6.1364179169700765 -0.774794 -24.3976 0 14 11 0.55 0.00 - yes Open
881 6.176569636524991 -0.838986 -26.0928 0 19 0 0.00 0.00 - yes Open
873 6.2987060644719 -0.84473 -26.2076 0 19 0 0.00 0.00 - yes Open
877 6.460596193474383 -0.823996 -25.8147 0 19 0 0.00 0.00 - yes Open
803 6.696921226225941 -0.778381 -24.3934 0 18 15 0.75 0.00 - yes Open
802 6.737152572584959 -0.80934 -24.9207 0 18 18 0.90 0.00 - yes Open
800 6.828955810971412 -0.797342 -23.8658 0 19 16 0.80 0.00 - yes Current
620 6.890565349006715 -0.992624 -28.6432 0 15 0 0.00 0.00 - yes Open
807 6.924363385512182 -0.789267 -24.8433 0 18 15 0.75 0.00 - yes Open
798 7.197254895005341 -0.83178 -25.6924 0 16 16 0.80 0.00 - yes Open
617 7.25695253679321 -0.943383 -24.9559 0 17 0 0.00 0.00 - yes Open
874 7.455804747405748 -0.790897 -20.6835 0 17 0 0.00 0.00 - yes Open
797 7.481414084461965 -0.82142 -26.2502 0 21 17 0.85 0.00 - yes Open
805 7.9142323766242315 -0.819836 -26.4257 0 21 17 0.85 0.00 - yes Open
884 55.83634397036696 -0.843594 -26.1424 0 18 0 0.00 0.00 - yes Open
616 56.02875660341615 -1.00343 -28.9633 0 15 0 0.00 0.00 - yes Open
619 56.83784189917394 -1.00164 -26.3548 0 15 0 0.00 0.00 - yes Open
804 57.194339723439576 -0.77967 -23.1691 0 19 16 0.80 0.00 - yes Open
612 57.4222504101707 -1.08289 -32.3895 1 17 0 0.00 0.00 - yes Open
799 57.975958599277476 -0.773564 -19.6304 0 18 15 0.75 0.00 - yes Open
875 58.73167053078245 -0.687968 -20.6455 0 18 0 0.00 0.00 - yes Open
808 58.975628311942216 -0.757633 -22.2892 0 18 15 0.75 0.00 - yes Open
879 59.98350652153543 -0.688332 -19.289 0 19 0 0.00 0.00 - yes Open

Molecular metrics

RDKit SASA burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -23.866kcal/mol
Ligand efficiency (LE) -0.7458kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -7.334
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 32HA

Physicochemical properties

Molecular weight 422.6Da
Lipinski: ≤ 500 Da
LogP (cLogP) 3.87
Lipinski: ≤ 5
Rotatable bonds 3

Conformational strain (MMFF94s)

Strain energy (ΔE) 19.15kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 154.64kcal/mol
Minimised FF energy 135.48kcal/mol

SASA & burial

not yet run
SASA has not been computed yet for this pose. Queue a background recompute to populate SASA burial metrics without blocking the page.