FAIRMol

Z56958949

Pose ID 3207 Compound 237 Pose 3207

DB Docking_panel_21Docking pose analysis is being read from this database.
Molecular metrics status: done
Cached molecular metrics are available for this pose.
Metrics cached · SASA missing
T02
Dihydrofolate reductase Homo sapiens
Ligand Z56958949
PDB5SD8

3D complex viewer

Strict H-bonds Permissive H-bonds
Viewer legend
Protein receptor
Pocket residues
Cofactor context
Docked ligand
Overall assessment
Reject No SASA yet
Promising but geometrically suspicious
Binding strong Geometry low Native mixed SASA missing
Strain ΔE
48.7 kcal/mol
Protein clashes
3
Internal clashes
3
Native overlap
contact recall 0.52, Jaccard 0.44, H-bond role recall 0.20
Burial
91%
Reason: strain 48.7 kcal/mol
strain ΔE 48.7 kcal/mol 3 protein-contact clashes 3 intramolecular clashes
Molecular report
Full metrics ↗
Reject Multiple quality flags — this pose should be deprioritised or discarded.
✓ Excellent LE (-0.558 kcal/mol/HA) ✓ Good fit quality (FQ -5.58) ✓ Good H-bonds (3 bonds) ✗ Extreme strain energy (48.7 kcal/mol) ✗ Geometry warnings ✗ Excluded by docking heuristics ℹ SASA not computed
Score
-18.974
kcal/mol
LE
-0.558
kcal/mol/HA
Fit Quality
-5.58
FQ (Leeson)
HAC
34
heavy atoms
MW
514
Da
LogP
2.43
cLogP
Strain ΔE
48.7 kcal/mol
SASA buried
computing…

Interaction summary

HB 3 HY 24 PI 2 CLASH 3
Final rank10.812Score-18.974
Inter norm-0.663Intra norm0.104
Top1000noExcludedyes
Contacts15H-bonds1
Artifact reasonexcluded; hard geometry fail; 1 severe clash; 1 protein clash; high strain Δ 61.1
Residues
ALA10 ARG29 ASN65 GLU31 ILE8 LEU23 LEU28 NAP201 PHE32 PHE35 PRO27 TRP25 TYR122 VAL116 VAL9

Protein summary

200 residues
Protein targetT02Atoms3128
Residues200Chains2
Residue summaryLYS:374; LEU:361; GLU:240; VAL:224; ARG:192; PHE:180; ILE:171; PRO:168; ASN:140; SER:132; TYR:126; GLN:119; ASP:108; MET:102; THR:98; GLY:91

Receptor context

1 kept / 0 excluded
Receptor context filtering: interactions and SASA are computed against protein atoms plus allowed cofactors/ions. Native ligand-like HETATM partners are excluded from scoring.
Kept context 1 Excluded HETATM 0
Kept cofactors / ions
A:NAP201

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: permissive.
Name5SD8Contacts21
PoseOpen native poseHB0
IFP residues
ALA10 ASN65 ASP22 GLN36 GLU31 GLY117 GLY21 ILE61 ILE8 LEU23 LEU68 NAP201 PHE32 PHE35 PRO62 SER60 THR137 THR57 TYR122 VAL116 VAL9
Current overlap11Native recall0.52
Jaccard0.44RMSD-
HB strict1Strict recall0.20
HB same residue+role1HB role recall0.20
HB same residue1HB residue recall0.20

HB · H-bonds

Mode: permissive. Count shows atom-level H-bonds; unique residues in summary: 0.

PI · π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

HY · Hydrophobic contacts

CLASH · Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBCTCT overlapCT recallHB role rec.RMSDExcluded
3206 4.948815307706374 -0.684734 -23.3162 1 18 17 0.81 0.00 - no Open
3703 5.418972328285989 -0.620116 -19.2603 3 17 0 0.00 0.00 - no Open
2378 8.222562756337524 -0.79336 -24.4281 7 17 0 0.00 0.00 - no Open
3702 7.61940434743973 -0.745467 -24.4793 4 14 0 0.00 0.00 - yes Open
2376 8.192807940647587 -0.845605 -25.0189 7 18 0 0.00 0.00 - yes Open
2379 10.032734323736642 -0.838117 -20.277 11 16 0 0.00 0.00 - yes Open
3207 10.811693932797503 -0.662537 -18.9743 1 15 11 0.52 0.20 - yes Current
3704 11.093703929308662 -0.700711 -22.7493 4 13 0 0.00 0.00 - yes Open
3205 11.162627935924707 -0.691385 -18.3515 4 19 15 0.71 0.00 - yes Open
3701 59.59594328498775 -0.634484 -20.5254 2 14 0 0.00 0.00 - yes Open
3204 60.01081702260929 -0.798969 -26.4833 1 19 18 0.86 0.00 - yes Open
2377 62.61832617806778 -0.717906 -21.9928 12 17 0 0.00 0.00 - yes Open

Molecular metrics

RDKit SASA burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -18.974kcal/mol
Ligand efficiency (LE) -0.5581kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -5.584
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 34HA

Physicochemical properties

Molecular weight 513.6Da
Lipinski: ≤ 500 Da
LogP (cLogP) 2.43
Lipinski: ≤ 5
Rotatable bonds 4

Conformational strain (MMFF94s)

Strain energy (ΔE) 48.73kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 48.32kcal/mol
Minimised FF energy -0.41kcal/mol

SASA & burial

not yet run
SASA has not been computed yet for this pose. Queue a background recompute to populate SASA burial metrics without blocking the page.