FAIRMol

OHD_TB2021_105

Pose ID 13074 Compound 1552 Pose 221

DB Docking_panel_21Docking pose analysis is being read from this database.
Molecular metrics status: done
Cached molecular metrics are available for this pose.
Metrics cached · SASA missing
T08
Pteridine reductase 1 (PTR1) Trypanosoma brucei
Ligand OHD_TB2021_105
PDB6RX6

3D complex viewer

Strict H-bonds Permissive H-bonds
Viewer legend
Protein receptor
Pocket residues
Cofactor context
Docked ligand
Overall assessment
Promising No SASA yet
Promising and worth follow-up
Binding strong Geometry high Native strong SASA missing
Strain ΔE
14.7 kcal/mol
Protein clashes
2
Internal clashes
2
Native overlap
contact recall 0.74, Jaccard 0.67, H-bond role recall 0.40
Burial
68%
Reason: no major geometry red flags detected
2 protein-contact clashes
Molecular report
Full metrics ↗
Promising Reasonable quality metrics. Warrants further investigation.
✓ Excellent LE (-1.319 kcal/mol/HA) ✓ Good fit quality (FQ -11.99) ✓ Strong H-bond network (6 bonds) ✗ Moderate strain (14.7 kcal/mol) ✗ Geometry warnings ✗ Minor protein-contact clashes (4) ✗ Internal clashes (9) ℹ SASA not computed
Score
-32.974
kcal/mol
LE
-1.319
kcal/mol/HA
Fit Quality
-11.99
FQ (Leeson)
HAC
25
heavy atoms
MW
340
Da
LogP
3.58
cLogP
Strain ΔE
14.7 kcal/mol
SASA buried
computing…

Interaction summary

HB 6 HY 17 PI 1 CLASH 2
Final rank2.295Score-32.974
Inter norm-1.405Intra norm0.086
Top1000noExcludedno
Contacts16H-bonds5
Artifact reasongeometry warning; 9 clashes; 4 protein contact clashes; moderate strain Δ 15.7
Residues
ARG14 ASP161 CYS168 GLY205 LEU208 LEU209 LYS13 LYS178 NAP301 PHE97 PRO210 SER207 TRP221 TYR174 VAL206 VAL211

Protein summary

258 residues
Protein targetT08Atoms3881
Residues258Chains2
Residue summaryLEU:437; VAL:433; ALA:361; ARG:288; ILE:266; GLU:210; LYS:198; SER:198; ASN:182; THR:154; GLN:153; PHE:140; PRO:140; TYR:126; GLY:112; HIS:103

Receptor context

1 kept / 0 excluded
Receptor context filtering: interactions and SASA are computed against protein atoms plus allowed cofactors/ions. Native ligand-like HETATM partners are excluded from scoring.
Kept context 1 Excluded HETATM 0
Kept cofactors / ions
A:NAP301

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: permissive.
NameTbPTR1_cW_6RX6_ReadyContacts19
PoseOpen native poseHB0
IFP residues
ARG14 ASP161 CYS168 GLY205 LEU208 LEU209 LYS178 MET213 NAP301 PHE171 PHE97 PRO210 PRO99 SER207 SER95 TRP221 TYR174 TYR98 VAL206
Current overlap14Native recall0.74
Jaccard0.67RMSD-
HB strict3Strict recall0.50
HB same residue+role2HB role recall0.40
HB same residue2HB residue recall0.40

HB · H-bonds

Mode: permissive. Count shows atom-level H-bonds; unique residues in summary: 0.

PI · π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

HY · Hydrophobic contacts

CLASH · Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBCTCT overlapCT recallHB role rec.RMSDExcluded
221 2.295370834023591 -1.40486 -32.9741 5 16 14 0.74 0.40 - no Current
222 4.5413919417840765 -1.16915 -26.6574 6 15 13 0.68 0.40 - yes Open

Molecular metrics

RDKit SASA burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -32.974kcal/mol
Ligand efficiency (LE) -1.3190kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -11.991
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 25HA

Physicochemical properties

Molecular weight 340.5Da
Lipinski: ≤ 500 Da
LogP (cLogP) 3.58
Lipinski: ≤ 5
Rotatable bonds 7

Conformational strain (MMFF94s)

Strain energy (ΔE) 14.71kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 37.11kcal/mol
Minimised FF energy 22.41kcal/mol

SASA & burial

not yet run
SASA has not been computed yet for this pose. Queue a background recompute to populate SASA burial metrics without blocking the page.