FAIRMol

Reverse docking explorer

Search one compound across many targets or scan the strongest compound-target pairs in the active database. The combined reverse-docking score uses a normalized docking-score estimator together with an interaction-fingerprint component.

DB fairmolExplorer results are being read from this database.
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1 compounds in matrix 8 best compound-target hits listed 8 targets
• Combined reverse-docking score = 65% normalized docking-score estimator + 35% interaction-fingerprint component.
• When a native ligand exists for an experiment, the interaction-fingerprint component is driven by similarity to the native contact/H-bond pattern.
• When no native ligand exists, the interaction-fingerprint component falls back to contact richness within the experiment (normalized contacts and H-bonds).

Compounds × targets matrix

Each cell shows the best combined reverse-docking score found for that compound on that target. Blank cells mean no imported pose passed the current filters.
Compound Best Mean Targets T01T03T05T07T08T09T14T20
Z57388199
[H]N(/N=C\c1c(C)nn(-c2ccccc2)c1C)C(=O)c1cc(-c2cccc3ccccc23)n([H])n1
0.926 0.827 8 0.84 0.82 0.87 0.84 0.93 0.79 0.76 0.76

Best compound-target hits

The score column is the combined reverse-docking score. The next two columns expose its components: normalized score-estimator and interaction fingerprint.
CompoundTargetExperimentCombinedScore partIFP partIFP modeMetricDock scoreInter normContactsHB
Z57388199
[H]N(/N=C\c1c(C)nn(-c2ccccc2)c1C)C(=O)c1cc(-c2cccc3ccccc23)n([H])n1
T08
native IFP available
T08
selection_import_t08
0.926 1.000 0.788 native_similarity final_rank_score -31.1583 -0.976286 18 10 Pose
Z57388199
[H]N(/N=C\c1c(C)nn(-c2ccccc2)c1C)C(=O)c1cc(-c2cccc3ccccc23)n([H])n1
T05
native IFP available
T05
selection_import_t05
0.867 1.000 0.620 native_similarity final_rank_score -27.3014 -0.885772 18 5 Pose
Z57388199
[H]N(/N=C\c1c(C)nn(-c2ccccc2)c1C)C(=O)c1cc(-c2cccc3ccccc23)n([H])n1
T07
native IFP available
T07
selection_import_t07
0.845 1.000 0.557 native_similarity final_rank_score -26.8898 -0.929769 16 1 Pose
Z57388199
[H]N(/N=C\c1c(C)nn(-c2ccccc2)c1C)C(=O)c1cc(-c2cccc3ccccc23)n([H])n1
T01
native IFP available
T01
selection_import_t01
0.844 1.000 0.555 native_similarity final_rank_score -27.1209 -0.813433 19 1 Pose
Z57388199
[H]N(/N=C\c1c(C)nn(-c2ccccc2)c1C)C(=O)c1cc(-c2cccc3ccccc23)n([H])n1
T03
native IFP available
T03
selection_import_t03
0.823 1.000 0.494 native_similarity final_rank_score -25.1232 -0.85665 19 3 Pose
Z57388199
[H]N(/N=C\c1c(C)nn(-c2ccccc2)c1C)C(=O)c1cc(-c2cccc3ccccc23)n([H])n1
T09
native IFP available
T09
selection_import_t09
0.792 1.000 0.406 native_similarity final_rank_score -21.8212 -0.869106 17 6 Pose
Z57388199
[H]N(/N=C\c1c(C)nn(-c2ccccc2)c1C)C(=O)c1cc(-c2cccc3ccccc23)n([H])n1
T20
native IFP available
T20
selection_import_t20
0.762 1.000 0.321 native_similarity final_rank_score -18.9765 -0.601271 12 5 Pose
Z57388199
[H]N(/N=C\c1c(C)nn(-c2ccccc2)c1C)C(=O)c1cc(-c2cccc3ccccc23)n([H])n1
T14
native IFP available
T14
selection_import_t14
0.760 1.000 0.313 native_similarity final_rank_score -18.7342 -0.677901 9 7 Pose