FAIRMol

Reverse docking explorer

Search one compound across many targets or scan the strongest compound-target pairs in the active database. The combined reverse-docking score uses a normalized docking-score estimator together with an interaction-fingerprint component.

DB fairmolExplorer results are being read from this database.
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2 compounds in matrix 6 best compound-target hits listed 6 targets
• Combined reverse-docking score = 65% normalized docking-score estimator + 35% interaction-fingerprint component.
• When a native ligand exists for an experiment, the interaction-fingerprint component is driven by similarity to the native contact/H-bond pattern.
• When no native ligand exists, the interaction-fingerprint component falls back to contact richness within the experiment (normalized contacts and H-bonds).

Compounds × targets matrix

Each cell shows the best combined reverse-docking score found for that compound on that target. Blank cells mean no imported pose passed the current filters.
Compound Best Mean Targets T03T04T05T11T18T22
Z56811592
[H]N([H])c1nnc(CCN2C(=O)S/C(=C/c3ccc(N(C)C)cc3)C2=O)s1
0.893 0.821 4 0.79 0.89 0.78 0.82
Z56811592
[H]N([H])c1nnc(CCN2C(=O)S/C(=C\c3ccc(N(C)C)cc3)C2=O)s1
0.847 0.826 2 0.85 0.80

Best compound-target hits

The score column is the combined reverse-docking score. The next two columns expose its components: normalized score-estimator and interaction fingerprint.
CompoundTargetExperimentCombinedScore partIFP partIFP modeMetricDock scoreInter normContactsHB
Z56811592
[H]N([H])c1nnc(CCN2C(=O)S/C(=C/c3ccc(N(C)C)cc3)C2=O)s1
T05
native IFP available
T05
selection_import_t05
0.893 1.000 0.695 native_similarity final_rank_score -33.3174 -1.18417 13 6 Pose
Z56811592
[H]N([H])c1nnc(CCN2C(=O)S/C(=C\c3ccc(N(C)C)cc3)C2=O)s1
T04
native IFP available
T04
selection_import_t04
0.847 1.000 0.562 native_similarity final_rank_score -28.5446 -1.08581 12 5 Pose
Z56811592
[H]N([H])c1nnc(CCN2C(=O)S/C(=C/c3ccc(N(C)C)cc3)C2=O)s1
T22
native IFP available
T22
selection_import_t22
0.815 1.000 0.473 native_similarity final_rank_score -31.5724 -1.24952 19 13 Pose
Z56811592
[H]N([H])c1nnc(CCN2C(=O)S/C(=C\c3ccc(N(C)C)cc3)C2=O)s1
T18
native IFP available
T18
selection_import_t18
0.804 1.000 0.441 native_similarity final_rank_score -25.4353 -0.975966 16 6 Pose
Z56811592
[H]N([H])c1nnc(CCN2C(=O)S/C(=C/c3ccc(N(C)C)cc3)C2=O)s1
T03
native IFP available
T03
selection_import_t03
0.793 1.000 0.408 native_similarity final_rank_score -28.5777 -1.08364 15 5 Pose
Z56811592
[H]N([H])c1nnc(CCN2C(=O)S/C(=C/c3ccc(N(C)C)cc3)C2=O)s1
T11
native IFP available
T11
selection_import_t11
0.782 1.000 0.378 native_similarity final_rank_score -22.1 -0.976606 21 6 Pose