FAIRMol

Reverse docking explorer

Search one compound across many targets or scan the strongest compound-target pairs in the active database. The combined reverse-docking score uses a normalized docking-score estimator together with an interaction-fingerprint component.

DB fairmolExplorer results are being read from this database.
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2 compounds in matrix 6 best compound-target hits listed 6 targets
• Combined reverse-docking score = 65% normalized docking-score estimator + 35% interaction-fingerprint component.
• When a native ligand exists for an experiment, the interaction-fingerprint component is driven by similarity to the native contact/H-bond pattern.
• When no native ligand exists, the interaction-fingerprint component falls back to contact richness within the experiment (normalized contacts and H-bonds).

Compounds × targets matrix

Each cell shows the best combined reverse-docking score found for that compound on that target. Blank cells mean no imported pose passed the current filters.
Compound Best Mean Targets T02T06T11T17T18T20
Z56798284
[H]Oc1c(/C=N/N=C(\O)c2cc(-c3ccc4ccccc4c3)nn2[H])cccc1CC=C
0.895 0.895 1 0.90
Z56798284
[H]Oc1c(/C=N\N([H])C(=O)c2cc(-c3ccc4ccccc4c3)nn2[H])cccc1CC=C
0.864 0.816 5 0.82 0.81 0.78 0.81 0.86

Best compound-target hits

The score column is the combined reverse-docking score. The next two columns expose its components: normalized score-estimator and interaction fingerprint.
CompoundTargetExperimentCombinedScore partIFP partIFP modeMetricDock scoreInter normContactsHB
Z56798284
[H]Oc1c(/C=N/N=C(\O)c2cc(-c3ccc4ccccc4c3)nn2[H])cccc1CC=C
T11
native IFP available
T11
selection_import_t11
0.895 1.000 0.701 native_similarity final_rank_score -22.0818 -0.824135 13 5 Pose
Z56798284
[H]Oc1c(/C=N\N([H])C(=O)c2cc(-c3ccc4ccccc4c3)nn2[H])cccc1CC=C
T20
native IFP available
T20
selection_import_t20
0.864 1.000 0.612 native_similarity final_rank_score -19.3115 -0.660659 13 7 Pose
Z56798284
[H]Oc1c(/C=N\N([H])C(=O)c2cc(-c3ccc4ccccc4c3)nn2[H])cccc1CC=C
T02
native IFP available
T02
selection_import_t02
0.820 1.000 0.485 native_similarity final_rank_score -21.9705 -0.84408 20 3 Pose
Z56798284
[H]Oc1c(/C=N\N([H])C(=O)c2cc(-c3ccc4ccccc4c3)nn2[H])cccc1CC=C
T06
native IFP available
T06
selection_import_t06
0.812 1.000 0.464 native_similarity final_rank_score -13.244 -0.83686 18 3 Pose
Z56798284
[H]Oc1c(/C=N\N([H])C(=O)c2cc(-c3ccc4ccccc4c3)nn2[H])cccc1CC=C
T18
native IFP available
T18
selection_import_t18
0.809 1.000 0.453 native_similarity final_rank_score -18.4215 -0.74441 15 2 Pose
Z56798284
[H]Oc1c(/C=N\N([H])C(=O)c2cc(-c3ccc4ccccc4c3)nn2[H])cccc1CC=C
T17
native IFP available
T17
selection_import_t17
0.776 1.000 0.360 native_similarity final_rank_score -19.9896 -0.756172 16 9 Pose