FAIRMol

Reverse docking explorer

Search one compound across many targets or scan the strongest compound-target pairs in the active database. The combined reverse-docking score uses a normalized docking-score estimator together with an interaction-fingerprint component.

DB fairmolExplorer results are being read from this database.
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4 compounds in matrix 4 best compound-target hits listed 4 targets
• Combined reverse-docking score = 65% normalized docking-score estimator + 35% interaction-fingerprint component.
• When a native ligand exists for an experiment, the interaction-fingerprint component is driven by similarity to the native contact/H-bond pattern.
• When no native ligand exists, the interaction-fingerprint component falls back to contact richness within the experiment (normalized contacts and H-bonds).

Compounds × targets matrix

Each cell shows the best combined reverse-docking score found for that compound on that target. Blank cells mean no imported pose passed the current filters.
Compound Best Mean Targets T04T05T10T19
Z49728506
C/C(=N/N=C(\O)[C@@H]1COc2ccccc2O1)c1ccccn1
0.859 0.859 1 0.86
Z49728506
C/C(=N/N=C(\O)[C@H]1COc2ccccc2O1)c1ccccn1
0.841 0.841 1 0.84
Z49728506
[H]N(/N=C(\C)c1ccccn1)C(=O)[C@H]1COc2ccccc2O1
0.800 0.800 1 0.80
Z49728506
C/C(=N\N=C(/O)[C@@H]1COc2ccccc2O1)c1ccccn1
0.726 0.726 1 0.73

Best compound-target hits

The score column is the combined reverse-docking score. The next two columns expose its components: normalized score-estimator and interaction fingerprint.
CompoundTargetExperimentCombinedScore partIFP partIFP modeMetricDock scoreInter normContactsHB
Z49728506
C/C(=N/N=C(\O)[C@@H]1COc2ccccc2O1)c1ccccn1
T10
native IFP available
T10
selection_import_t10
0.859 1.000 0.597 native_similarity final_rank_score -23.5496 -1.10349 13 14 Pose
Z49728506
C/C(=N/N=C(\O)[C@H]1COc2ccccc2O1)c1ccccn1
T05
native IFP available
T05
selection_import_t05
0.841 1.000 0.547 native_similarity final_rank_score -29.8772 -1.29721 12 6 Pose
Z49728506
[H]N(/N=C(\C)c1ccccn1)C(=O)[C@H]1COc2ccccc2O1
T04
native IFP available
T04
selection_import_t04
0.800 1.000 0.428 native_similarity final_rank_score -23.4562 -1.08518 10 1 Pose
Z49728506
C/C(=N\N=C(/O)[C@@H]1COc2ccccc2O1)c1ccccn1
T19
native IFP available
T19
selection_import_t19
0.726 1.000 0.218 native_similarity final_rank_score -31.4514 -1.41092 17 7 Pose