FAIRMol

Reverse docking explorer

Search one compound across many targets or scan the strongest compound-target pairs in the active database. The combined reverse-docking score uses a normalized docking-score estimator together with an interaction-fingerprint component.

DB fairmolExplorer results are being read from this database.
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2 compounds in matrix 5 best compound-target hits listed 5 targets
• Combined reverse-docking score = 65% normalized docking-score estimator + 35% interaction-fingerprint component.
• When a native ligand exists for an experiment, the interaction-fingerprint component is driven by similarity to the native contact/H-bond pattern.
• When no native ligand exists, the interaction-fingerprint component falls back to contact richness within the experiment (normalized contacts and H-bonds).

Compounds × targets matrix

Each cell shows the best combined reverse-docking score found for that compound on that target. Blank cells mean no imported pose passed the current filters.
Compound Best Mean Targets T06T12T16T17T22
Z1924722291
[H]n1nc(C[C@@H]2CCN(C(=O)C3CC3)C2)n(-c2ccc(-c3ccc4occc4c3)cc2)c1=O
0.869 0.835 4 0.83 0.85 0.79 0.87
Z1924722291
[H]n1nc(O)[n+](-c2ccc(-c3ccc4occc4c3)cc2)c1C[C@@H]1CCN(C(=O)C2CC2)C1
0.795 0.795 1 0.80

Best compound-target hits

The score column is the combined reverse-docking score. The next two columns expose its components: normalized score-estimator and interaction fingerprint.
CompoundTargetExperimentCombinedScore partIFP partIFP modeMetricDock scoreInter normContactsHB
Z1924722291
[H]n1nc(C[C@@H]2CCN(C(=O)C3CC3)C2)n(-c2ccc(-c3ccc4occc4c3)cc2)c1=O
T22
native IFP available
T22
selection_import_t22
0.869 1.000 0.627 native_similarity final_rank_score -28.8552 -0.963441 22 8 Pose
Z1924722291
[H]n1nc(C[C@@H]2CCN(C(=O)C3CC3)C2)n(-c2ccc(-c3ccc4occc4c3)cc2)c1=O
T12
native IFP available
T12
selection_import_t12
0.850 1.000 0.571 native_similarity final_rank_score -31.2866 -0.856142 18 9 Pose
Z1924722291
[H]n1nc(C[C@@H]2CCN(C(=O)C3CC3)C2)n(-c2ccc(-c3ccc4occc4c3)cc2)c1=O
T06
native IFP available
T06
selection_import_t06
0.834 1.000 0.526 native_similarity final_rank_score -26.2714 -0.837146 20 2 Pose
Z1924722291
[H]n1nc(O)[n+](-c2ccc(-c3ccc4occc4c3)cc2)c1C[C@@H]1CCN(C(=O)C2CC2)C1
T16
native IFP available
T16
selection_import_t16
0.795 1.000 0.414 native_similarity final_rank_score -24.2755 -0.729871 16 3 Pose
Z1924722291
[H]n1nc(C[C@@H]2CCN(C(=O)C3CC3)C2)n(-c2ccc(-c3ccc4occc4c3)cc2)c1=O
T17
native IFP available
T17
selection_import_t17
0.786 1.000 0.389 native_similarity final_rank_score -24.6647 -0.726559 19 5 Pose