FAIRMol

Reverse docking explorer

Search one compound across many targets or scan the strongest compound-target pairs in the active database. The combined reverse-docking score uses a normalized docking-score estimator together with an interaction-fingerprint component.

DB fairmolExplorer results are being read from this database.
Reset
2 compounds in matrix 2 best compound-target hits listed 2 targets
• Combined reverse-docking score = 65% normalized docking-score estimator + 35% interaction-fingerprint component.
• When a native ligand exists for an experiment, the interaction-fingerprint component is driven by similarity to the native contact/H-bond pattern.
• When no native ligand exists, the interaction-fingerprint component falls back to contact richness within the experiment (normalized contacts and H-bonds).

Compounds × targets matrix

Each cell shows the best combined reverse-docking score found for that compound on that target. Blank cells mean no imported pose passed the current filters.
Compound Best Mean Targets T15T16
OSA_Lib_264
[H][N+]1(C)CCN(CC(=O)N2C[C@H]3[C@@H](c4ccccc4)C[C@]([N+]4([H])CCCC4)(C[C@@H]3c3ccccc3)C2)CC1
0.852 0.852 1 0.85
OSA_Lib_264
[H][N+]1(CC(=O)N2C[C@@H]3[C@@H](c4ccccc4)C[C@@]([N+]4([H])CCCC4)(C[C@H]3c3ccccc3)C2)CCN(C)CC1
0.766 0.766 1 0.77

Best compound-target hits

The score column is the combined reverse-docking score. The next two columns expose its components: normalized score-estimator and interaction fingerprint.
CompoundTargetExperimentCombinedScore partIFP partIFP modeMetricDock scoreInter normContactsHB
OSA_Lib_264
[H][N+]1(C)CCN(CC(=O)N2C[C@H]3[C@@H](c4ccccc4)C[C@]([N+]4([H])CCCC4)(C[C@@H]3c3ccccc3)C2)CC1
T15
native IFP available
T15
selection_import_t15
0.852 1.000 0.577 native_similarity final_rank_score -24.0953 -0.68486 15 2 Pose
OSA_Lib_264
[H][N+]1(CC(=O)N2C[C@@H]3[C@@H](c4ccccc4)C[C@@]([N+]4([H])CCCC4)(C[C@H]3c3ccccc3)C2)CCN(C)CC1
T16
native IFP available
T16
selection_import_t16
0.766 1.000 0.331 native_similarity final_rank_score -22.2947 -0.659609 13 2 Pose