FAIRMol

Reverse docking explorer

Search one compound across many targets or scan the strongest compound-target pairs in the active database. The combined reverse-docking score uses a normalized docking-score estimator together with an interaction-fingerprint component.

DB fairmolExplorer results are being read from this database.
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1 compounds in matrix 13 best compound-target hits listed 13 targets
• Combined reverse-docking score = 65% normalized docking-score estimator + 35% interaction-fingerprint component.
• When a native ligand exists for an experiment, the interaction-fingerprint component is driven by similarity to the native contact/H-bond pattern.
• When no native ligand exists, the interaction-fingerprint component falls back to contact richness within the experiment (normalized contacts and H-bonds).

Compounds × targets matrix

Each cell shows the best combined reverse-docking score found for that compound on that target. Blank cells mean no imported pose passed the current filters.
Compound Best Mean Targets T01T03T05T07T08T09T10T12T13T15T17T18T22
OHD_MAC_75
[H]Oc1cc(/C=N/N([H])c2ncnc3c(N([H])c4ccc(OC)cc4)ncnc23)ccc1O
0.910 0.845 13 0.86 0.84 0.84 0.89 0.82 0.80 0.89 0.91 0.87 0.80 0.74 0.82 0.90

Best compound-target hits

The score column is the combined reverse-docking score. The next two columns expose its components: normalized score-estimator and interaction fingerprint.
CompoundTargetExperimentCombinedScore partIFP partIFP modeMetricDock scoreInter normContactsHB
OHD_MAC_75
[H]Oc1cc(/C=N/N([H])c2ncnc3c(N([H])c4ccc(OC)cc4)ncnc23)ccc1O
T12
native IFP available
T12
selection_import_t12
0.910 1.000 0.744 native_similarity final_rank_score -24.1715 -1.03956 16 10 Pose
OHD_MAC_75
[H]Oc1cc(/C=N/N([H])c2ncnc3c(N([H])c4ccc(OC)cc4)ncnc23)ccc1O
T22
native IFP available
T22
selection_import_t22
0.905 1.000 0.728 native_similarity final_rank_score -26.8884 -1.11238 23 10 Pose
OHD_MAC_75
[H]Oc1cc(/C=N/N([H])c2ncnc3c(N([H])c4ccc(OC)cc4)ncnc23)ccc1O
T07
native IFP available
T07
selection_import_t07
0.891 1.000 0.690 native_similarity final_rank_score -24.053 -1.02007 18 9 Pose
OHD_MAC_75
[H]Oc1cc(/C=N/N([H])c2ncnc3c(N([H])c4ccc(OC)cc4)ncnc23)ccc1O
T10
native IFP available
T10
selection_import_t10
0.887 1.000 0.677 native_similarity final_rank_score -14.126 -0.80723 18 13 Pose
OHD_MAC_75
[H]Oc1cc(/C=N/N([H])c2ncnc3c(N([H])c4ccc(OC)cc4)ncnc23)ccc1O
T13
native IFP available
T13
selection_import_t13
0.868 1.000 0.623 native_similarity final_rank_score -25.9132 -1.04489 24 11 Pose
OHD_MAC_75
[H]Oc1cc(/C=N/N([H])c2ncnc3c(N([H])c4ccc(OC)cc4)ncnc23)ccc1O
T01
native IFP available
T01
selection_import_t01
0.859 1.000 0.599 native_similarity final_rank_score -23.6453 -0.873051 19 4 Pose
OHD_MAC_75
[H]Oc1cc(/C=N/N([H])c2ncnc3c(N([H])c4ccc(OC)cc4)ncnc23)ccc1O
T05
native IFP available
T05
selection_import_t05
0.841 1.000 0.547 native_similarity final_rank_score -28.6013 -1.03868 16 9 Pose
OHD_MAC_75
[H]Oc1cc(/C=N/N([H])c2ncnc3c(N([H])c4ccc(OC)cc4)ncnc23)ccc1O
T03
native IFP available
T03
selection_import_t03
0.841 1.000 0.546 native_similarity final_rank_score -18.7883 -0.906801 18 7 Pose
OHD_MAC_75
[H]Oc1cc(/C=N/N([H])c2ncnc3c(N([H])c4ccc(OC)cc4)ncnc23)ccc1O
T18
native IFP available
T18
selection_import_t18
0.824 1.000 0.498 native_similarity final_rank_score -16.3353 -0.749474 16 9 Pose
OHD_MAC_75
[H]Oc1cc(/C=N/N([H])c2ncnc3c(N([H])c4ccc(OC)cc4)ncnc23)ccc1O
T08
native IFP available
T08
selection_import_t08
0.819 1.000 0.483 native_similarity final_rank_score -30.2922 -1.12038 18 6 Pose
OHD_MAC_75
[H]Oc1cc(/C=N/N([H])c2ncnc3c(N([H])c4ccc(OC)cc4)ncnc23)ccc1O
T15
native IFP available
T15
selection_import_t15
0.801 1.000 0.431 native_similarity final_rank_score -22.5539 -0.803675 17 5 Pose
OHD_MAC_75
[H]Oc1cc(/C=N/N([H])c2ncnc3c(N([H])c4ccc(OC)cc4)ncnc23)ccc1O
T09
native IFP available
T09
selection_import_t09
0.799 1.000 0.426 native_similarity final_rank_score -24.7512 -0.892376 16 6 Pose
OHD_MAC_75
[H]Oc1cc(/C=N/N([H])c2ncnc3c(N([H])c4ccc(OC)cc4)ncnc23)ccc1O
T17
native IFP available
T17
selection_import_t17
0.739 1.000 0.254 native_similarity final_rank_score -20.3167 -0.781705 17 7 Pose