FAIRMol

Reverse docking explorer

Search one compound across many targets or scan the strongest compound-target pairs in the active database. The combined reverse-docking score uses a normalized docking-score estimator together with an interaction-fingerprint component.

DB fairmolExplorer results are being read from this database.
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2 compounds in matrix 7 best compound-target hits listed 7 targets
• Combined reverse-docking score = 65% normalized docking-score estimator + 35% interaction-fingerprint component.
• When a native ligand exists for an experiment, the interaction-fingerprint component is driven by similarity to the native contact/H-bond pattern.
• When no native ligand exists, the interaction-fingerprint component falls back to contact richness within the experiment (normalized contacts and H-bonds).

Compounds × targets matrix

Each cell shows the best combined reverse-docking score found for that compound on that target. Blank cells mean no imported pose passed the current filters.
Compound Best Mean Targets T03T11T13T15T17T19T20
OHD_Babesia_23
[H]OCCN(C)CCN(C)c1ccc(/N=C/C=[N+](/C)CCO[H])c2c1C(=O)c1c(O[H])ccc(O[H])c1C2=O
0.922 0.922 1 0.92
OHD_Babesia_23
[H]OCC/[N+](C)=C/C=N\c1ccc(N(C)CC[N@+]([H])(C)CCO[H])c2c1C(=O)c1c(O[H])ccc(O[H])c1C2=O
0.863 0.814 6 0.82 0.85 0.86 0.80 0.84 0.71

Best compound-target hits

The score column is the combined reverse-docking score. The next two columns expose its components: normalized score-estimator and interaction fingerprint.
CompoundTargetExperimentCombinedScore partIFP partIFP modeMetricDock scoreInter normContactsHB
OHD_Babesia_23
[H]OCCN(C)CCN(C)c1ccc(/N=C/C=[N+](/C)CCO[H])c2c1C(=O)c1c(O[H])ccc(O[H])c1C2=O
T20
native IFP available
T20
selection_import_t20
0.922 1.000 0.778 native_similarity final_rank_score -18.5622 -0.575628 12 5 Pose
OHD_Babesia_23
[H]OCC/[N+](C)=C/C=N\c1ccc(N(C)CC[N@+]([H])(C)CCO[H])c2c1C(=O)c1c(O[H])ccc(O[H])c1C2=O
T13
native IFP available
T13
selection_import_t13
0.863 1.000 0.609 native_similarity final_rank_score -17.9408 -0.803277 22 10 Pose
OHD_Babesia_23
[H]OCC/[N+](C)=C/C=N\c1ccc(N(C)CC[N@+]([H])(C)CCO[H])c2c1C(=O)c1c(O[H])ccc(O[H])c1C2=O
T11
native IFP available
T11
selection_import_t11
0.849 1.000 0.570 native_similarity final_rank_score -19.3464 -0.720357 16 9 Pose
OHD_Babesia_23
[H]OCC/[N+](C)=C/C=N\c1ccc(N(C)CC[N@+]([H])(C)CCO[H])c2c1C(=O)c1c(O[H])ccc(O[H])c1C2=O
T17
native IFP available
T17
selection_import_t17
0.843 1.000 0.553 native_similarity final_rank_score -22.2462 -0.659197 19 8 Pose
OHD_Babesia_23
[H]OCC/[N+](C)=C/C=N\c1ccc(N(C)CC[N@+]([H])(C)CCO[H])c2c1C(=O)c1c(O[H])ccc(O[H])c1C2=O
T03
native IFP available
T03
selection_import_t03
0.820 1.000 0.485 native_similarity final_rank_score -24.9885 -0.809493 20 5 Pose
OHD_Babesia_23
[H]OCC/[N+](C)=C/C=N\c1ccc(N(C)CC[N@+]([H])(C)CCO[H])c2c1C(=O)c1c(O[H])ccc(O[H])c1C2=O
T15
native IFP available
T15
selection_import_t15
0.801 1.000 0.431 native_similarity final_rank_score -19.2853 -0.669361 17 7 Pose
OHD_Babesia_23
[H]OCC/[N+](C)=C/C=N\c1ccc(N(C)CC[N@+]([H])(C)CCO[H])c2c1C(=O)c1c(O[H])ccc(O[H])c1C2=O
T19
native IFP available
T19
selection_import_t19
0.708 1.000 0.167 native_similarity final_rank_score -26.0699 -0.901719 22 10 Pose