FAIRMol

Reverse docking explorer

Search one compound across many targets or scan the strongest compound-target pairs in the active database. The combined reverse-docking score uses a normalized docking-score estimator together with an interaction-fingerprint component.

DB fairmolExplorer results are being read from this database.
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1 compounds in matrix 6 best compound-target hits listed 6 targets
• Combined reverse-docking score = 65% normalized docking-score estimator + 35% interaction-fingerprint component.
• When a native ligand exists for an experiment, the interaction-fingerprint component is driven by similarity to the native contact/H-bond pattern.
• When no native ligand exists, the interaction-fingerprint component falls back to contact richness within the experiment (normalized contacts and H-bonds).

Compounds × targets matrix

Each cell shows the best combined reverse-docking score found for that compound on that target. Blank cells mean no imported pose passed the current filters.
Compound Best Mean Targets T01T02T03T15T17T19
MK190
[H]OCc1ccc(Cl)c(C(=O)N([H])CC2(COc3ccc(-c4cc(=S)ss4)cc3)CCCCC2)c1
0.931 0.828 6 0.81 0.81 0.93 0.78 0.93 0.72

Best compound-target hits

The score column is the combined reverse-docking score. The next two columns expose its components: normalized score-estimator and interaction fingerprint.
CompoundTargetExperimentCombinedScore partIFP partIFP modeMetricDock scoreInter normContactsHB
MK190
[H]OCc1ccc(Cl)c(C(=O)N([H])CC2(COc3ccc(-c4cc(=S)ss4)cc3)CCCCC2)c1
T03
native IFP available
T03
selection_import_t03
0.931 1.000 0.804 native_similarity final_rank_score -25.8454 -0.816947 19 6 Pose
MK190
[H]OCc1ccc(Cl)c(C(=O)N([H])CC2(COc3ccc(-c4cc(=S)ss4)cc3)CCCCC2)c1
T17
native IFP available
T17
selection_import_t17
0.928 1.000 0.795 native_similarity final_rank_score -23.9654 -0.740468 19 3 Pose
MK190
[H]OCc1ccc(Cl)c(C(=O)N([H])CC2(COc3ccc(-c4cc(=S)ss4)cc3)CCCCC2)c1
T02
native IFP available
T02
selection_import_t02
0.809 1.000 0.454 native_similarity final_rank_score -24.6404 -0.781101 19 2 Pose
MK190
[H]OCc1ccc(Cl)c(C(=O)N([H])CC2(COc3ccc(-c4cc(=S)ss4)cc3)CCCCC2)c1
T01
native IFP available
T01
selection_import_t01
0.805 1.000 0.443 native_similarity final_rank_score -28.4152 -0.802507 16 2 Pose
MK190
[H]OCc1ccc(Cl)c(C(=O)N([H])CC2(COc3ccc(-c4cc(=S)ss4)cc3)CCCCC2)c1
T15
native IFP available
T15
selection_import_t15
0.780 1.000 0.371 native_similarity final_rank_score -14.874 -0.72292 18 3 Pose
MK190
[H]OCc1ccc(Cl)c(C(=O)N([H])CC2(COc3ccc(-c4cc(=S)ss4)cc3)CCCCC2)c1
T19
native IFP available
T19
selection_import_t19
0.717 1.000 0.190 native_similarity final_rank_score -27.9485 -0.967782 22 4 Pose