FAIRMol

Reverse docking explorer

Search one compound across many targets or scan the strongest compound-target pairs in the active database. The combined reverse-docking score uses a normalized docking-score estimator together with an interaction-fingerprint component.

DB fairmolExplorer results are being read from this database.
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2 compounds in matrix 3 best compound-target hits listed 3 targets
• Combined reverse-docking score = 65% normalized docking-score estimator + 35% interaction-fingerprint component.
• When a native ligand exists for an experiment, the interaction-fingerprint component is driven by similarity to the native contact/H-bond pattern.
• When no native ligand exists, the interaction-fingerprint component falls back to contact richness within the experiment (normalized contacts and H-bonds).

Compounds × targets matrix

Each cell shows the best combined reverse-docking score found for that compound on that target. Blank cells mean no imported pose passed the current filters.
Compound Best Mean Targets T08T18T19
KB_Leish_37
[H]N([H])c1nc(N([H])[H])[n+]([H])c2nc(-c3cccc4ccccc34)cc(C)c12
0.868 0.815 2 0.87 0.76
KB_Leish_37
[H]N([H])c1nc(N([H])[H])c2c(C)cc(-c3cccc4ccccc34)nc2n1
0.734 0.734 1 0.73

Best compound-target hits

The score column is the combined reverse-docking score. The next two columns expose its components: normalized score-estimator and interaction fingerprint.
CompoundTargetExperimentCombinedScore partIFP partIFP modeMetricDock scoreInter normContactsHB
KB_Leish_37
[H]N([H])c1nc(N([H])[H])[n+]([H])c2nc(-c3cccc4ccccc34)cc(C)c12
T08
native IFP available
T08
selection_import_t08
0.868 1.000 0.622 native_similarity final_rank_score -33.5676 -1.45258 16 7 Pose
KB_Leish_37
[H]N([H])c1nc(N([H])[H])[n+]([H])c2nc(-c3cccc4ccccc34)cc(C)c12
T18
native IFP available
T18
selection_import_t18
0.763 1.000 0.323 native_similarity final_rank_score -21.1476 -0.89539 6 2 Pose
KB_Leish_37
[H]N([H])c1nc(N([H])[H])c2c(C)cc(-c3cccc4ccccc34)nc2n1
T19
native IFP available
T19
selection_import_t19
0.734 1.000 0.240 native_similarity final_rank_score -31.976 -1.39463 18 5 Pose