FAIRMol

Reverse docking explorer

Search one compound across many targets or scan the strongest compound-target pairs in the active database. The combined reverse-docking score uses a normalized docking-score estimator together with an interaction-fingerprint component.

DB fairmolExplorer results are being read from this database.
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1 compounds in matrix 3 best compound-target hits listed 3 targets
• Combined reverse-docking score = 65% normalized docking-score estimator + 35% interaction-fingerprint component.
• When a native ligand exists for an experiment, the interaction-fingerprint component is driven by similarity to the native contact/H-bond pattern.
• When no native ligand exists, the interaction-fingerprint component falls back to contact richness within the experiment (normalized contacts and H-bonds).

Compounds × targets matrix

Each cell shows the best combined reverse-docking score found for that compound on that target. Blank cells mean no imported pose passed the current filters.
Compound Best Mean Targets T02T14T21
KB_HAT_132
[H]OC[C@H](c1ccccc1)N([H])c1nccc(-c2c(-c3ccc(F)cc3)ncn2C2CC[N+]([H])([H])CC2)n1
0.858 0.810 3 0.86 0.75 0.82

Best compound-target hits

The score column is the combined reverse-docking score. The next two columns expose its components: normalized score-estimator and interaction fingerprint.
CompoundTargetExperimentCombinedScore partIFP partIFP modeMetricDock scoreInter normContactsHB
KB_HAT_132
[H]OC[C@H](c1ccccc1)N([H])c1nccc(-c2c(-c3ccc(F)cc3)ncn2C2CC[N+]([H])([H])CC2)n1
T02
native IFP available
T02
selection_import_t02
0.858 1.000 0.595 native_similarity final_rank_score -23.1277 -0.83894 17 6 Pose
KB_HAT_132
[H]OC[C@H](c1ccccc1)N([H])c1nccc(-c2c(-c3ccc(F)cc3)ncn2C2CC[N+]([H])([H])CC2)n1
T21
native IFP available
T21
selection_import_t21
0.821 1.000 0.487 native_similarity final_rank_score -23.1494 -0.772708 11 8 Pose
KB_HAT_132
[H]OC[C@H](c1ccccc1)N([H])c1nccc(-c2c(-c3ccc(F)cc3)ncn2C2CC[N+]([H])([H])CC2)n1
T14
native IFP available
T14
selection_import_t14
0.751 1.000 0.288 native_similarity final_rank_score -23.3116 -0.655069 18 5 Pose