FAIRMol

Reverse docking explorer

Search one compound across many targets or scan the strongest compound-target pairs in the active database. The combined reverse-docking score uses a normalized docking-score estimator together with an interaction-fingerprint component.

DB fairmolExplorer results are being read from this database.
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1 compounds in matrix 7 best compound-target hits listed 7 targets
• Combined reverse-docking score = 65% normalized docking-score estimator + 35% interaction-fingerprint component.
• When a native ligand exists for an experiment, the interaction-fingerprint component is driven by similarity to the native contact/H-bond pattern.
• When no native ligand exists, the interaction-fingerprint component falls back to contact richness within the experiment (normalized contacts and H-bonds).

Compounds × targets matrix

Each cell shows the best combined reverse-docking score found for that compound on that target. Blank cells mean no imported pose passed the current filters.
Compound Best Mean Targets T01T02T06T07T08T11T18
KB_HAT_118
[H]N([H])C(=O)c1ncc(N([H])[C@@H]2CCC[N+]([H])([H])C2)nc1N([H])c1cccc(Cl)c1
0.887 0.838 7 0.85 0.88 0.82 0.89 0.83 0.81 0.79

Best compound-target hits

The score column is the combined reverse-docking score. The next two columns expose its components: normalized score-estimator and interaction fingerprint.
CompoundTargetExperimentCombinedScore partIFP partIFP modeMetricDock scoreInter normContactsHB
KB_HAT_118
[H]N([H])C(=O)c1ncc(N([H])[C@@H]2CCC[N+]([H])([H])C2)nc1N([H])c1cccc(Cl)c1
T07
native IFP available
T07
selection_import_t07
0.887 1.000 0.677 native_similarity final_rank_score -35.3362 -1.33485 16 9 Pose
KB_HAT_118
[H]N([H])C(=O)c1ncc(N([H])[C@@H]2CCC[N+]([H])([H])C2)nc1N([H])c1cccc(Cl)c1
T02
native IFP available
T02
selection_import_t02
0.879 1.000 0.655 native_similarity final_rank_score -22.1541 -1.08501 17 4 Pose
KB_HAT_118
[H]N([H])C(=O)c1ncc(N([H])[C@@H]2CCC[N+]([H])([H])C2)nc1N([H])c1cccc(Cl)c1
T01
native IFP available
T01
selection_import_t01
0.851 1.000 0.574 native_similarity final_rank_score -25.2784 -1.06423 19 6 Pose
KB_HAT_118
[H]N([H])C(=O)c1ncc(N([H])[C@@H]2CCC[N+]([H])([H])C2)nc1N([H])c1cccc(Cl)c1
T08
native IFP available
T08
selection_import_t08
0.833 1.000 0.523 native_similarity final_rank_score -22.4311 -1.35753 13 12 Pose
KB_HAT_118
[H]N([H])C(=O)c1ncc(N([H])[C@@H]2CCC[N+]([H])([H])C2)nc1N([H])c1cccc(Cl)c1
T06
native IFP available
T06
selection_import_t06
0.816 1.000 0.475 native_similarity final_rank_score -22.7934 -0.980685 17 4 Pose
KB_HAT_118
[H]N([H])C(=O)c1ncc(N([H])[C@@H]2CCC[N+]([H])([H])C2)nc1N([H])c1cccc(Cl)c1
T11
native IFP available
T11
selection_import_t11
0.813 1.000 0.465 native_similarity final_rank_score -19.4856 -1.01212 18 4 Pose
KB_HAT_118
[H]N([H])C(=O)c1ncc(N([H])[C@@H]2CCC[N+]([H])([H])C2)nc1N([H])c1cccc(Cl)c1
T18
native IFP available
T18
selection_import_t18
0.789 1.000 0.397 native_similarity final_rank_score -11.2779 -0.89686 15 5 Pose