FAIRMol

Reverse docking explorer

Search one compound across many targets or scan the strongest compound-target pairs in the active database. The combined reverse-docking score uses a normalized docking-score estimator together with an interaction-fingerprint component.

DB fairmolExplorer results are being read from this database.
Reset
1 compounds in matrix 7 best compound-target hits listed 7 targets
• Combined reverse-docking score = 65% normalized docking-score estimator + 35% interaction-fingerprint component.
• When a native ligand exists for an experiment, the interaction-fingerprint component is driven by similarity to the native contact/H-bond pattern.
• When no native ligand exists, the interaction-fingerprint component falls back to contact richness within the experiment (normalized contacts and H-bonds).

Compounds × targets matrix

Each cell shows the best combined reverse-docking score found for that compound on that target. Blank cells mean no imported pose passed the current filters.
Compound Best Mean Targets T01T02T10T11T17T19T22
KB_HAT_115
[H]N([H])C(=O)c1ccccc1N([H])c1nc(N([H])[C@H]2CC[C@H](N([H])S(C)(=O)=O)CC2)ncc1Br
0.952 0.855 7 0.84 0.92 0.95 0.89 0.75 0.73 0.90

Best compound-target hits

The score column is the combined reverse-docking score. The next two columns expose its components: normalized score-estimator and interaction fingerprint.
CompoundTargetExperimentCombinedScore partIFP partIFP modeMetricDock scoreInter normContactsHB
KB_HAT_115
[H]N([H])C(=O)c1ccccc1N([H])c1nc(N([H])[C@H]2CC[C@H](N([H])S(C)(=O)=O)CC2)ncc1Br
T10
native IFP available
T10
selection_import_t10
0.952 1.000 0.864 native_similarity final_rank_score -13.2707 -0.942215 17 11 Pose
KB_HAT_115
[H]N([H])C(=O)c1ccccc1N([H])c1nc(N([H])[C@H]2CC[C@H](N([H])S(C)(=O)=O)CC2)ncc1Br
T02
native IFP available
T02
selection_import_t02
0.920 1.000 0.770 native_similarity final_rank_score -23.6644 -1.00152 20 6 Pose
KB_HAT_115
[H]N([H])C(=O)c1ccccc1N([H])c1nc(N([H])[C@H]2CC[C@H](N([H])S(C)(=O)=O)CC2)ncc1Br
T22
native IFP available
T22
selection_import_t22
0.904 1.000 0.726 native_similarity final_rank_score -24.6608 -1.05438 20 6 Pose
KB_HAT_115
[H]N([H])C(=O)c1ccccc1N([H])c1nc(N([H])[C@H]2CC[C@H](N([H])S(C)(=O)=O)CC2)ncc1Br
T11
native IFP available
T11
selection_import_t11
0.893 1.000 0.695 native_similarity final_rank_score -19.1155 -0.847649 17 5 Pose
KB_HAT_115
[H]N([H])C(=O)c1ccccc1N([H])c1nc(N([H])[C@H]2CC[C@H](N([H])S(C)(=O)=O)CC2)ncc1Br
T01
native IFP available
T01
selection_import_t01
0.837 1.000 0.535 native_similarity final_rank_score -19.2987 -0.987041 17 7 Pose
KB_HAT_115
[H]N([H])C(=O)c1ccccc1N([H])c1nc(N([H])[C@H]2CC[C@H](N([H])S(C)(=O)=O)CC2)ncc1Br
T17
native IFP available
T17
selection_import_t17
0.748 1.000 0.279 native_similarity final_rank_score -18.5212 -0.90859 22 8 Pose
KB_HAT_115
[H]N([H])C(=O)c1ccccc1N([H])c1nc(N([H])[C@H]2CC[C@H](N([H])S(C)(=O)=O)CC2)ncc1Br
T19
native IFP available
T19
selection_import_t19
0.731 1.000 0.232 native_similarity final_rank_score -30.6381 -1.07485 22 7 Pose