FAIRMol

Reverse docking explorer

Search one compound across many targets or scan the strongest compound-target pairs in the active database. The combined reverse-docking score uses a normalized docking-score estimator together with an interaction-fingerprint component.

DB fairmolExplorer results are being read from this database.
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2 compounds in matrix 3 best compound-target hits listed 3 targets
• Combined reverse-docking score = 65% normalized docking-score estimator + 35% interaction-fingerprint component.
• When a native ligand exists for an experiment, the interaction-fingerprint component is driven by similarity to the native contact/H-bond pattern.
• When no native ligand exists, the interaction-fingerprint component falls back to contact richness within the experiment (normalized contacts and H-bonds).

Compounds × targets matrix

Each cell shows the best combined reverse-docking score found for that compound on that target. Blank cells mean no imported pose passed the current filters.
Compound Best Mean Targets T04T07T18
CKP-39
[H]N([H])c1ccc2c(c1)ncn2Cc1ccc2ccccc2c1
0.834 0.796 2 0.83 0.76
CKP-39
[H]N([H])c1ccc2c(c1)[n+]([H])cn2Cc1ccc2ccccc2c1
0.821 0.821 1 0.82

Best compound-target hits

The score column is the combined reverse-docking score. The next two columns expose its components: normalized score-estimator and interaction fingerprint.
CompoundTargetExperimentCombinedScore partIFP partIFP modeMetricDock scoreInter normContactsHB
CKP-39
[H]N([H])c1ccc2c(c1)ncn2Cc1ccc2ccccc2c1
T04
native IFP available
T04
selection_import_t04
0.834 1.000 0.525 native_similarity final_rank_score -26.0093 -1.2555 11 2 Pose
CKP-39
[H]N([H])c1ccc2c(c1)[n+]([H])cn2Cc1ccc2ccccc2c1
T07
native IFP available
T07
selection_import_t07
0.821 1.000 0.489 native_similarity final_rank_score -29.8942 -1.45619 13 6 Pose
CKP-39
[H]N([H])c1ccc2c(c1)ncn2Cc1ccc2ccccc2c1
T18
native IFP available
T18
selection_import_t18
0.758 1.000 0.309 native_similarity final_rank_score -20.1775 -0.979973 13 2 Pose