FAIRMol

Reverse docking explorer

Search one compound across many targets or scan the strongest compound-target pairs in the active database. The combined reverse-docking score uses a normalized docking-score estimator together with an interaction-fingerprint component.

DB SELECTIONExplorer results are being read from this database.
Reset
1 compounds in matrix 5 best compound-target hits listed 5 targets
• Combined reverse-docking score = 65% normalized docking-score estimator + 35% interaction-fingerprint component.
• When a native ligand exists for an experiment, the interaction-fingerprint component is driven by similarity to the native contact/H-bond pattern.
• When no native ligand exists, the interaction-fingerprint component falls back to contact richness within the experiment (normalized contacts and H-bonds).

Compounds × targets matrix

Each cell shows the best combined reverse-docking score found for that compound on that target. Blank cells mean no imported pose passed the current filters.
Compound Best Mean Targets T04T07T08T14T18
Z57781571
[H]Oc1ccc(/C=N\N=c2/sc(N([H])C(C)=O)c(-c3ccc(C)cc3)n2[H])cc1
0.875 0.821 5 0.82 0.87 0.85 0.78 0.77

Best compound-target hits

The score column is the combined reverse-docking score. The next two columns expose its components: normalized score-estimator and interaction fingerprint.
CompoundTargetExperimentCombinedScore partIFP partIFP modeMetricDock scoreInter normContactsHB
Z57781571
[H]Oc1ccc(/C=N\N=c2/sc(N([H])C(C)=O)c(-c3ccc(C)cc3)n2[H])cc1
T07
native IFP available
T07
selection_import_t07
0.875 1.000 0.643 native_similarity final_rank_score -28.6007 -1.199 17 6 Pose
Z57781571
[H]Oc1ccc(/C=N\N=c2/sc(N([H])C(C)=O)c(-c3ccc(C)cc3)n2[H])cc1
T08
native IFP available
T08
selection_import_t08
0.851 1.000 0.574 native_similarity final_rank_score -31.7101 -1.21926 12 7 Pose
Z57781571
[H]Oc1ccc(/C=N\N=c2/sc(N([H])C(C)=O)c(-c3ccc(C)cc3)n2[H])cc1
T04
native IFP available
T04
selection_import_t04
0.821 1.000 0.489 native_similarity final_rank_score -20.9222 -0.929712 13 3 Pose
Z57781571
[H]Oc1ccc(/C=N\N=c2/sc(N([H])C(C)=O)c(-c3ccc(C)cc3)n2[H])cc1
T14
native IFP available
T14
selection_import_t14
0.784 1.000 0.382 native_similarity final_rank_score -21.5818 -0.875522 15 6 Pose
Z57781571
[H]Oc1ccc(/C=N\N=c2/sc(N([H])C(C)=O)c(-c3ccc(C)cc3)n2[H])cc1
T18
native IFP available
T18
selection_import_t18
0.774 1.000 0.353 native_similarity final_rank_score -21.0438 -0.871034 14 5 Pose