FAIRMol

Reverse docking explorer

Search one compound across many targets or scan the strongest compound-target pairs in the active database. The combined reverse-docking score uses a normalized docking-score estimator together with an interaction-fingerprint component.

DB SELECTIONExplorer results are being read from this database.
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3 compounds in matrix 4 best compound-target hits listed 4 targets
• Combined reverse-docking score = 65% normalized docking-score estimator + 35% interaction-fingerprint component.
• When a native ligand exists for an experiment, the interaction-fingerprint component is driven by similarity to the native contact/H-bond pattern.
• When no native ligand exists, the interaction-fingerprint component falls back to contact richness within the experiment (normalized contacts and H-bonds).

Compounds × targets matrix

Each cell shows the best combined reverse-docking score found for that compound on that target. Blank cells mean no imported pose passed the current filters.
Compound Best Mean Targets T01T09T13T14
Z49894254
[H]n1c[n+]([H])/c(=N\[N+]([H])=C/c2ccc(C(C)C)cc2)c2c3c(sc21)CCCC3
0.879 0.817 2 0.88 0.76
Z49894254
[H]N(/N=C\c1ccc(C(C)C)cc1)c1ncnc2sc3c(c12)CCCC3
0.869 0.869 1 0.87
Z49894254
[H]n1c[n+]([H])/c(=N\[N+]([H])=C\c2ccc(C(C)C)cc2)c2c3c(sc21)CCCC3
0.778 0.778 1 0.78

Best compound-target hits

The score column is the combined reverse-docking score. The next two columns expose its components: normalized score-estimator and interaction fingerprint.
CompoundTargetExperimentCombinedScore partIFP partIFP modeMetricDock scoreInter normContactsHB
Z49894254
[H]n1c[n+]([H])/c(=N\[N+]([H])=C/c2ccc(C(C)C)cc2)c2c3c(sc21)CCCC3
T01
native IFP available
T01
selection_import_t01
0.879 1.000 0.653 native_similarity final_rank_score -24.9833 -1.0578 16 3 Pose
Z49894254
[H]N(/N=C\c1ccc(C(C)C)cc1)c1ncnc2sc3c(c12)CCCC3
T13
native IFP available
T13
selection_import_t13
0.869 1.000 0.624 native_similarity final_rank_score -30.775 -1.11692 15 8 Pose
Z49894254
[H]n1c[n+]([H])/c(=N\[N+]([H])=C\c2ccc(C(C)C)cc2)c2c3c(sc21)CCCC3
T14
native IFP available
T14
selection_import_t14
0.778 1.000 0.365 native_similarity final_rank_score -19.49 -0.918311 15 3 Pose
Z49894254
[H]n1c[n+]([H])/c(=N\[N+]([H])=C/c2ccc(C(C)C)cc2)c2c3c(sc21)CCCC3
T09
native IFP available
T09
selection_import_t09
0.756 1.000 0.303 native_similarity final_rank_score -22.7587 -1.07471 14 5 Pose