FAIRMol

Reverse docking explorer

Search one compound across many targets or scan the strongest compound-target pairs in the active database. The combined reverse-docking score uses a normalized docking-score estimator together with an interaction-fingerprint component.

DB SELECTIONExplorer results are being read from this database.
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4 compounds in matrix 21 best compound-target hits listed 21 targets
• Combined reverse-docking score = 65% normalized docking-score estimator + 35% interaction-fingerprint component.
• When a native ligand exists for an experiment, the interaction-fingerprint component is driven by similarity to the native contact/H-bond pattern.
• When no native ligand exists, the interaction-fingerprint component falls back to contact richness within the experiment (normalized contacts and H-bonds).

Compounds × targets matrix

Each cell shows the best combined reverse-docking score found for that compound on that target. Blank cells mean no imported pose passed the current filters.
Compound Best Mean Targets T01T03T04T05T06T07T08T09T10T11T12T13T14T15T16T17T18T19T20T21T22
Z44831771
[H]Oc1ccc(O[H])c(/C(C)=N\N([H])c2cccc(/C(O)=N/N=C(\C)c3cc(O[H])ccc3O[H])c2)c1
0.925 0.890 5 0.86 0.89 0.93 0.87 0.91
Z44831771
[H]Oc1ccc(O[H])c(/C(C)=N\N=C(/O)c2cccc(N([H])/N=C(\C)c3cc(O[H])ccc3O[H])c2)c1
0.917 0.851 6 0.84 0.86 0.89 0.92 0.80 0.79
Z44831771
[H]Oc1ccc(O[H])c(/C(C)=N/Nc2cccc(C(=O)N([H])/N=C(\C)c3cc(O[H])ccc3O[H])c2)c1
0.904 0.855 8 0.88 0.90 0.89 0.75 0.80 0.82 0.89 0.90
Z44831771
[H]Oc1ccc(O[H])c(/C(C)=N\N=C(/O)c2cccc(N([H])/N=C(/C)c3cc(O[H])ccc3O[H])c2)c1
0.839 0.822 2 0.84 0.81

Best compound-target hits

The score column is the combined reverse-docking score. The next two columns expose its components: normalized score-estimator and interaction fingerprint.
CompoundTargetExperimentCombinedScore partIFP partIFP modeMetricDock scoreInter normContactsHB
Z44831771
[H]Oc1ccc(O[H])c(/C(C)=N\N([H])c2cccc(/C(O)=N/N=C(\C)c3cc(O[H])ccc3O[H])c2)c1
T10
native IFP available
T10
selection_import_t10
0.925 1.000 0.787 native_similarity final_rank_score -27.4463 -0.798482 20 12 Pose
Z44831771
[H]Oc1ccc(O[H])c(/C(C)=N\N=C(/O)c2cccc(N([H])/N=C(\C)c3cc(O[H])ccc3O[H])c2)c1
T11
native IFP available
T11
selection_import_t11
0.917 1.000 0.763 native_similarity final_rank_score -27.0912 -0.884359 15 5 Pose
Z44831771
[H]Oc1ccc(O[H])c(/C(C)=N\N([H])c2cccc(/C(O)=N/N=C(\C)c3cc(O[H])ccc3O[H])c2)c1
T22
native IFP available
T22
selection_import_t22
0.911 1.000 0.745 native_similarity final_rank_score -26.665 -1.03902 22 14 Pose
Z44831771
[H]Oc1ccc(O[H])c(/C(C)=N/Nc2cccc(C(=O)N([H])/N=C(\C)c3cc(O[H])ccc3O[H])c2)c1
T21
native IFP available
T21
selection_import_t21
0.904 1.000 0.726 native_similarity final_rank_score -34.7577 -0.941146 18 14 Pose
Z44831771
[H]Oc1ccc(O[H])c(/C(C)=N/Nc2cccc(C(=O)N([H])/N=C(\C)c3cc(O[H])ccc3O[H])c2)c1
T04
native IFP available
T04
selection_import_t04
0.901 1.000 0.716 native_similarity final_rank_score -30.879 -0.942522 14 7 Pose
Z44831771
[H]Oc1ccc(O[H])c(/C(C)=N/Nc2cccc(C(=O)N([H])/N=C(\C)c3cc(O[H])ccc3O[H])c2)c1
T12
native IFP available
T12
selection_import_t12
0.894 1.000 0.697 native_similarity final_rank_score -30.7908 -1.04701 18 11 Pose
Z44831771
[H]Oc1ccc(O[H])c(/C(C)=N\N=C(/O)c2cccc(N([H])/N=C(\C)c3cc(O[H])ccc3O[H])c2)c1
T09
native IFP available
T09
selection_import_t09
0.893 1.000 0.695 native_similarity final_rank_score -31.1008 -1.07835 19 9 Pose
Z44831771
[H]Oc1ccc(O[H])c(/C(C)=N/Nc2cccc(C(=O)N([H])/N=C(\C)c3cc(O[H])ccc3O[H])c2)c1
T20
native IFP available
T20
selection_import_t20
0.890 1.000 0.685 native_similarity final_rank_score -21.3543 -0.748819 13 7 Pose
Z44831771
[H]Oc1ccc(O[H])c(/C(C)=N\N([H])c2cccc(/C(O)=N/N=C(\C)c3cc(O[H])ccc3O[H])c2)c1
T07
native IFP available
T07
selection_import_t07
0.885 1.000 0.673 native_similarity final_rank_score -36.6574 -1.02054 15 8 Pose
Z44831771
[H]Oc1ccc(O[H])c(/C(C)=N/Nc2cccc(C(=O)N([H])/N=C(\C)c3cc(O[H])ccc3O[H])c2)c1
T01
native IFP available
T01
selection_import_t01
0.883 1.000 0.665 native_similarity final_rank_score -28.9224 -1.00427 20 7 Pose
Z44831771
[H]Oc1ccc(O[H])c(/C(C)=N\N([H])c2cccc(/C(O)=N/N=C(\C)c3cc(O[H])ccc3O[H])c2)c1
T13
native IFP available
T13
selection_import_t13
0.874 1.000 0.639 native_similarity final_rank_score -27.3542 -0.983333 22 13 Pose
Z44831771
[H]Oc1ccc(O[H])c(/C(C)=N\N=C(/O)c2cccc(N([H])/N=C(\C)c3cc(O[H])ccc3O[H])c2)c1
T08
native IFP available
T08
selection_import_t08
0.864 1.000 0.611 native_similarity final_rank_score -33.4208 -1.12559 17 9 Pose
Z44831771
[H]Oc1ccc(O[H])c(/C(C)=N\N([H])c2cccc(/C(O)=N/N=C(\C)c3cc(O[H])ccc3O[H])c2)c1
T06
native IFP available
T06
selection_import_t06
0.856 1.000 0.590 native_similarity final_rank_score -23.302 -0.789482 21 8 Pose
Z44831771
[H]Oc1ccc(O[H])c(/C(C)=N\N=C(/O)c2cccc(N([H])/N=C(\C)c3cc(O[H])ccc3O[H])c2)c1
T05
native IFP available
T05
selection_import_t05
0.841 1.000 0.547 native_similarity final_rank_score -33.8225 -1.08514 16 10 Pose
Z44831771
[H]Oc1ccc(O[H])c(/C(C)=N\N=C(/O)c2cccc(N([H])/N=C(/C)c3cc(O[H])ccc3O[H])c2)c1
T03
native IFP available
T03
selection_import_t03
0.839 1.000 0.541 native_similarity final_rank_score -32.7618 -1.18447 16 8 Pose
Z44831771
[H]Oc1ccc(O[H])c(/C(C)=N/Nc2cccc(C(=O)N([H])/N=C(\C)c3cc(O[H])ccc3O[H])c2)c1
T19
native IFP available
T19
selection_import_t19
0.823 1.000 0.494 native_similarity final_rank_score -29.2761 -1.03419 15 14 Pose
Z44831771
[H]Oc1ccc(O[H])c(/C(C)=N\N=C(/O)c2cccc(N([H])/N=C(/C)c3cc(O[H])ccc3O[H])c2)c1
T14
native IFP available
T14
selection_import_t14
0.805 1.000 0.444 native_similarity final_rank_score -26.4589 -0.766451 16 11 Pose
Z44831771
[H]Oc1ccc(O[H])c(/C(C)=N/Nc2cccc(C(=O)N([H])/N=C(\C)c3cc(O[H])ccc3O[H])c2)c1
T17
native IFP available
T17
selection_import_t17
0.798 1.000 0.424 native_similarity final_rank_score -26.8801 -0.947279 21 11 Pose
Z44831771
[H]Oc1ccc(O[H])c(/C(C)=N\N=C(/O)c2cccc(N([H])/N=C(\C)c3cc(O[H])ccc3O[H])c2)c1
T15
native IFP available
T15
selection_import_t15
0.797 1.000 0.419 native_similarity final_rank_score -22.6215 -0.851297 13 8 Pose
Z44831771
[H]Oc1ccc(O[H])c(/C(C)=N\N=C(/O)c2cccc(N([H])/N=C(\C)c3cc(O[H])ccc3O[H])c2)c1
T18
native IFP available
T18
selection_import_t18
0.793 1.000 0.408 native_similarity final_rank_score -17.9665 -0.829169 14 4 Pose
Z44831771
[H]Oc1ccc(O[H])c(/C(C)=N/Nc2cccc(C(=O)N([H])/N=C(\C)c3cc(O[H])ccc3O[H])c2)c1
T16
native IFP available
T16
selection_import_t16
0.747 1.000 0.276 native_similarity final_rank_score -33.8612 -0.859572 13 8 Pose