FAIRMol

Reverse docking explorer

Search one compound across many targets or scan the strongest compound-target pairs in the active database. The combined reverse-docking score uses a normalized docking-score estimator together with an interaction-fingerprint component.

DB SELECTIONExplorer results are being read from this database.
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2 compounds in matrix 6 best compound-target hits listed 6 targets
• Combined reverse-docking score = 65% normalized docking-score estimator + 35% interaction-fingerprint component.
• When a native ligand exists for an experiment, the interaction-fingerprint component is driven by similarity to the native contact/H-bond pattern.
• When no native ligand exists, the interaction-fingerprint component falls back to contact richness within the experiment (normalized contacts and H-bonds).

Compounds × targets matrix

Each cell shows the best combined reverse-docking score found for that compound on that target. Blank cells mean no imported pose passed the current filters.
Compound Best Mean Targets T05T08T11T14T15T22
Z24304592
[H]N([H])/C(C)=C(/C#N)C(=O)CSc1nc2scc(-c3ccccc3)c2c(=O)n1C
0.870 0.849 4 0.87 0.82 0.85 0.86
Z24304592
[H]N([H])/C(C)=C(\C#N)C(=O)CSc1nc2scc(-c3ccccc3)c2c(=O)n1C
0.806 0.790 2 0.81 0.77

Best compound-target hits

The score column is the combined reverse-docking score. The next two columns expose its components: normalized score-estimator and interaction fingerprint.
CompoundTargetExperimentCombinedScore partIFP partIFP modeMetricDock scoreInter normContactsHB
Z24304592
[H]N([H])/C(C)=C(/C#N)C(=O)CSc1nc2scc(-c3ccccc3)c2c(=O)n1C
T05
native IFP available
T05
selection_import_t05
0.870 1.000 0.627 native_similarity final_rank_score -29.5116 -1.08393 14 6 Pose
Z24304592
[H]N([H])/C(C)=C(/C#N)C(=O)CSc1nc2scc(-c3ccccc3)c2c(=O)n1C
T22
native IFP available
T22
selection_import_t22
0.857 1.000 0.591 native_similarity final_rank_score -32.1344 -1.15688 20 11 Pose
Z24304592
[H]N([H])/C(C)=C(/C#N)C(=O)CSc1nc2scc(-c3ccccc3)c2c(=O)n1C
T11
native IFP available
T11
selection_import_t11
0.847 1.000 0.563 native_similarity final_rank_score -24.9148 -0.888421 19 5 Pose
Z24304592
[H]N([H])/C(C)=C(/C#N)C(=O)CSc1nc2scc(-c3ccccc3)c2c(=O)n1C
T08
native IFP available
T08
selection_import_t08
0.823 1.000 0.494 native_similarity final_rank_score -32.1453 -1.22174 14 6 Pose
Z24304592
[H]N([H])/C(C)=C(\C#N)C(=O)CSc1nc2scc(-c3ccccc3)c2c(=O)n1C
T14
native IFP available
T14
selection_import_t14
0.806 1.000 0.447 native_similarity final_rank_score -24.385 -0.887855 19 7 Pose
Z24304592
[H]N([H])/C(C)=C(\C#N)C(=O)CSc1nc2scc(-c3ccccc3)c2c(=O)n1C
T15
native IFP available
T15
selection_import_t15
0.774 1.000 0.353 native_similarity final_rank_score -20.5563 -0.869958 14 4 Pose