FAIRMol

Reverse docking explorer

Search one compound across many targets or scan the strongest compound-target pairs in the active database. The combined reverse-docking score uses a normalized docking-score estimator together with an interaction-fingerprint component.

DB SELECTIONExplorer results are being read from this database.
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1 compounds in matrix 15 best compound-target hits listed 15 targets
• Combined reverse-docking score = 65% normalized docking-score estimator + 35% interaction-fingerprint component.
• When a native ligand exists for an experiment, the interaction-fingerprint component is driven by similarity to the native contact/H-bond pattern.
• When no native ligand exists, the interaction-fingerprint component falls back to contact richness within the experiment (normalized contacts and H-bonds).

Compounds × targets matrix

Each cell shows the best combined reverse-docking score found for that compound on that target. Blank cells mean no imported pose passed the current filters.
Compound Best Mean Targets T02T03T04T05T07T09T10T11T12T13T14T17T18T20T21
Z20255081
[H]Oc1ccc(C(=O)CSc2nnc(CSc3nc4ccccc4s3)n2CC)cc1O[H]
0.943 0.841 15 0.84 0.78 0.80 0.86 0.84 0.76 0.92 0.89 0.94 0.88 0.75 0.79 0.82 0.83 0.90

Best compound-target hits

The score column is the combined reverse-docking score. The next two columns expose its components: normalized score-estimator and interaction fingerprint.
CompoundTargetExperimentCombinedScore partIFP partIFP modeMetricDock scoreInter normContactsHB
Z20255081
[H]Oc1ccc(C(=O)CSc2nnc(CSc3nc4ccccc4s3)n2CC)cc1O[H]
T12
native IFP available
T12
selection_import_t12
0.943 1.000 0.836 native_similarity final_rank_score -29.8157 -1.15443 17 14 Pose
Z20255081
[H]Oc1ccc(C(=O)CSc2nnc(CSc3nc4ccccc4s3)n2CC)cc1O[H]
T10
native IFP available
T10
selection_import_t10
0.917 1.000 0.763 native_similarity final_rank_score -20.4087 -0.857475 15 13 Pose
Z20255081
[H]Oc1ccc(C(=O)CSc2nnc(CSc3nc4ccccc4s3)n2CC)cc1O[H]
T21
native IFP available
T21
selection_import_t21
0.896 1.000 0.704 native_similarity final_rank_score -21.9132 -0.886151 18 8 Pose
Z20255081
[H]Oc1ccc(C(=O)CSc2nnc(CSc3nc4ccccc4s3)n2CC)cc1O[H]
T11
native IFP available
T11
selection_import_t11
0.885 1.000 0.672 native_similarity final_rank_score -21.2615 -0.833689 15 10 Pose
Z20255081
[H]Oc1ccc(C(=O)CSc2nnc(CSc3nc4ccccc4s3)n2CC)cc1O[H]
T13
native IFP available
T13
selection_import_t13
0.884 1.000 0.669 native_similarity final_rank_score -24.0255 -0.944403 19 6 Pose
Z20255081
[H]Oc1ccc(C(=O)CSc2nnc(CSc3nc4ccccc4s3)n2CC)cc1O[H]
T05
native IFP available
T05
selection_import_t05
0.863 1.000 0.610 native_similarity final_rank_score -27.5305 -0.97422 15 8 Pose
Z20255081
[H]Oc1ccc(C(=O)CSc2nnc(CSc3nc4ccccc4s3)n2CC)cc1O[H]
T02
native IFP available
T02
selection_import_t02
0.845 1.000 0.557 native_similarity final_rank_score -25.5218 -0.989236 21 1 Pose
Z20255081
[H]Oc1ccc(C(=O)CSc2nnc(CSc3nc4ccccc4s3)n2CC)cc1O[H]
T07
native IFP available
T07
selection_import_t07
0.843 1.000 0.551 native_similarity final_rank_score -34.8331 -1.19533 17 9 Pose
Z20255081
[H]Oc1ccc(C(=O)CSc2nnc(CSc3nc4ccccc4s3)n2CC)cc1O[H]
T20
native IFP available
T20
selection_import_t20
0.831 1.000 0.517 native_similarity final_rank_score -17.4537 -0.65996 10 6 Pose
Z20255081
[H]Oc1ccc(C(=O)CSc2nnc(CSc3nc4ccccc4s3)n2CC)cc1O[H]
T18
native IFP available
T18
selection_import_t18
0.824 1.000 0.498 native_similarity final_rank_score -19.9579 -0.707052 16 8 Pose
Z20255081
[H]Oc1ccc(C(=O)CSc2nnc(CSc3nc4ccccc4s3)n2CC)cc1O[H]
T04
native IFP available
T04
selection_import_t04
0.800 1.000 0.429 native_similarity final_rank_score -24.243 -0.839972 13 2 Pose
Z20255081
[H]Oc1ccc(C(=O)CSc2nnc(CSc3nc4ccccc4s3)n2CC)cc1O[H]
T17
native IFP available
T17
selection_import_t17
0.789 1.000 0.396 native_similarity final_rank_score -22.0828 -0.896028 18 6 Pose
Z20255081
[H]Oc1ccc(C(=O)CSc2nnc(CSc3nc4ccccc4s3)n2CC)cc1O[H]
T03
native IFP available
T03
selection_import_t03
0.784 1.000 0.384 native_similarity final_rank_score -22.7906 -0.986403 13 5 Pose
Z20255081
[H]Oc1ccc(C(=O)CSc2nnc(CSc3nc4ccccc4s3)n2CC)cc1O[H]
T09
native IFP available
T09
selection_import_t09
0.756 1.000 0.303 native_similarity final_rank_score -23.8867 -0.894601 14 4 Pose
Z20255081
[H]Oc1ccc(C(=O)CSc2nnc(CSc3nc4ccccc4s3)n2CC)cc1O[H]
T14
native IFP available
T14
selection_import_t14
0.750 1.000 0.284 native_similarity final_rank_score -18.2749 -0.781192 14 8 Pose