FAIRMol

Reverse docking explorer

Search one compound across many targets or scan the strongest compound-target pairs in the active database. The combined reverse-docking score uses a normalized docking-score estimator together with an interaction-fingerprint component.

DB SELECTIONExplorer results are being read from this database.
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2 compounds in matrix 5 best compound-target hits listed 5 targets
• Combined reverse-docking score = 65% normalized docking-score estimator + 35% interaction-fingerprint component.
• When a native ligand exists for an experiment, the interaction-fingerprint component is driven by similarity to the native contact/H-bond pattern.
• When no native ligand exists, the interaction-fingerprint component falls back to contact richness within the experiment (normalized contacts and H-bonds).

Compounds × targets matrix

Each cell shows the best combined reverse-docking score found for that compound on that target. Blank cells mean no imported pose passed the current filters.
Compound Best Mean Targets T04T06T18T19T21
Z16382127
[H]N(C(=O)CSc1ncnc2c1cnn2-c1ccccc1)[C@H]1CCS(=O)(=O)C1
0.940 0.815 4 0.80 0.78 0.74 0.94
Z16382127
[H]N(C(=O)CSc1ncnc2c1cnn2-c1ccccc1)[C@@H]1CCS(=O)(=O)C1
0.827 0.827 1 0.83

Best compound-target hits

The score column is the combined reverse-docking score. The next two columns expose its components: normalized score-estimator and interaction fingerprint.
CompoundTargetExperimentCombinedScore partIFP partIFP modeMetricDock scoreInter normContactsHB
Z16382127
[H]N(C(=O)CSc1ncnc2c1cnn2-c1ccccc1)[C@H]1CCS(=O)(=O)C1
T21
native IFP available
T21
selection_import_t21
0.940 1.000 0.828 native_similarity final_rank_score -25.6343 -0.914349 16 14 Pose
Z16382127
[H]N(C(=O)CSc1ncnc2c1cnn2-c1ccccc1)[C@@H]1CCS(=O)(=O)C1
T06
native IFP available
T06
selection_import_t06
0.827 1.000 0.507 native_similarity final_rank_score -26.9951 -0.926626 18 2 Pose
Z16382127
[H]N(C(=O)CSc1ncnc2c1cnn2-c1ccccc1)[C@H]1CCS(=O)(=O)C1
T04
native IFP available
T04
selection_import_t04
0.805 1.000 0.442 native_similarity final_rank_score -27.529 -0.912628 12 0 Pose
Z16382127
[H]N(C(=O)CSc1ncnc2c1cnn2-c1ccccc1)[C@H]1CCS(=O)(=O)C1
T18
native IFP available
T18
selection_import_t18
0.777 1.000 0.362 native_similarity final_rank_score -25.5464 -0.859465 13 4 Pose
Z16382127
[H]N(C(=O)CSc1ncnc2c1cnn2-c1ccccc1)[C@H]1CCS(=O)(=O)C1
T19
native IFP available
T19
selection_import_t19
0.740 1.000 0.258 native_similarity final_rank_score -33.7196 -1.18678 17 6 Pose