FAIRMol

Reverse docking explorer

Search one compound across many targets or scan the strongest compound-target pairs in the active database. The combined reverse-docking score uses a normalized docking-score estimator together with an interaction-fingerprint component.

DB SELECTIONExplorer results are being read from this database.
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2 compounds in matrix 7 best compound-target hits listed 7 targets
• Combined reverse-docking score = 65% normalized docking-score estimator + 35% interaction-fingerprint component.
• When a native ligand exists for an experiment, the interaction-fingerprint component is driven by similarity to the native contact/H-bond pattern.
• When no native ligand exists, the interaction-fingerprint component falls back to contact richness within the experiment (normalized contacts and H-bonds).

Compounds × targets matrix

Each cell shows the best combined reverse-docking score found for that compound on that target. Blank cells mean no imported pose passed the current filters.
Compound Best Mean Targets T04T05T06T09T11T13T14
TC553
[H]N(Cc1cn([H])c2nc(N([H])C3CC3)ccc12)C(=O)c1cncc(C(=O)O)n1
0.872 0.841 3 0.87 0.87 0.78
TC553
[H]N(Cc1cn([H])c2c1ccc(N([H])C1CC1)[n+]2[H])C(=O)c1cncc(C(=O)O)n1
0.854 0.826 4 0.81 0.85 0.83 0.81

Best compound-target hits

The score column is the combined reverse-docking score. The next two columns expose its components: normalized score-estimator and interaction fingerprint.
CompoundTargetExperimentCombinedScore partIFP partIFP modeMetricDock scoreInter normContactsHB
TC553
[H]N(Cc1cn([H])c2nc(N([H])C3CC3)ccc12)C(=O)c1cncc(C(=O)O)n1
T04
native IFP available
T04
selection_import_t04
0.872 1.000 0.634 native_similarity final_rank_score -26.699 -0.951665 12 7 Pose
TC553
[H]N(Cc1cn([H])c2nc(N([H])C3CC3)ccc12)C(=O)c1cncc(C(=O)O)n1
T11
native IFP available
T11
selection_import_t11
0.867 1.000 0.620 native_similarity final_rank_score -20.9812 -0.92782 14 6 Pose
TC553
[H]N(Cc1cn([H])c2c1ccc(N([H])C1CC1)[n+]2[H])C(=O)c1cncc(C(=O)O)n1
T06
native IFP available
T06
selection_import_t06
0.854 1.000 0.582 native_similarity final_rank_score -26.7043 -0.952461 18 2 Pose
TC553
[H]N(Cc1cn([H])c2c1ccc(N([H])C1CC1)[n+]2[H])C(=O)c1cncc(C(=O)O)n1
T09
native IFP available
T09
selection_import_t09
0.833 1.000 0.524 native_similarity final_rank_score -28.7216 -1.15484 18 6 Pose
TC553
[H]N(Cc1cn([H])c2c1ccc(N([H])C1CC1)[n+]2[H])C(=O)c1cncc(C(=O)O)n1
T05
native IFP available
T05
selection_import_t05
0.809 1.000 0.454 native_similarity final_rank_score -25.997 -1.12186 12 12 Pose
TC553
[H]N(Cc1cn([H])c2c1ccc(N([H])C1CC1)[n+]2[H])C(=O)c1cncc(C(=O)O)n1
T13
native IFP available
T13
selection_import_t13
0.806 1.000 0.446 native_similarity final_rank_score -28.8816 -1.07479 16 10 Pose
TC553
[H]N(Cc1cn([H])c2nc(N([H])C3CC3)ccc12)C(=O)c1cncc(C(=O)O)n1
T14
native IFP available
T14
selection_import_t14
0.783 1.000 0.380 native_similarity final_rank_score -25.3995 -0.929915 13 6 Pose