FAIRMol

Reverse docking explorer

Search one compound across many targets or scan the strongest compound-target pairs in the active database. The combined reverse-docking score uses a normalized docking-score estimator together with an interaction-fingerprint component.

DB SELECTIONExplorer results are being read from this database.
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2 compounds in matrix 3 best compound-target hits listed 3 targets
• Combined reverse-docking score = 65% normalized docking-score estimator + 35% interaction-fingerprint component.
• When a native ligand exists for an experiment, the interaction-fingerprint component is driven by similarity to the native contact/H-bond pattern.
• When no native ligand exists, the interaction-fingerprint component falls back to contact richness within the experiment (normalized contacts and H-bonds).

Compounds × targets matrix

Each cell shows the best combined reverse-docking score found for that compound on that target. Blank cells mean no imported pose passed the current filters.
Compound Best Mean Targets T05T06T09
TC428
[H]N(Cc1cn([H])c2c1ccc(N([H])C1CC1)[n+]2[H])C(=O)c1nccc(C(=O)O)n1
0.872 0.840 2 0.81 0.87
TC428
[H]N(Cc1cn([H])c2nc(N([H])C3CC3)ccc12)C(=O)c1nccc(C(=O)O)n1
0.843 0.843 1 0.84

Best compound-target hits

The score column is the combined reverse-docking score. The next two columns expose its components: normalized score-estimator and interaction fingerprint.
CompoundTargetExperimentCombinedScore partIFP partIFP modeMetricDock scoreInter normContactsHB
TC428
[H]N(Cc1cn([H])c2c1ccc(N([H])C1CC1)[n+]2[H])C(=O)c1nccc(C(=O)O)n1
T09
native IFP available
T09
selection_import_t09
0.872 1.000 0.633 native_similarity final_rank_score -22.2334 -0.983257 17 7 Pose
TC428
[H]N(Cc1cn([H])c2nc(N([H])C3CC3)ccc12)C(=O)c1nccc(C(=O)O)n1
T06
native IFP available
T06
selection_import_t06
0.843 1.000 0.550 native_similarity final_rank_score -16.029 -0.992154 17 3 Pose
TC428
[H]N(Cc1cn([H])c2c1ccc(N([H])C1CC1)[n+]2[H])C(=O)c1nccc(C(=O)O)n1
T05
native IFP available
T05
selection_import_t05
0.809 1.000 0.454 native_similarity final_rank_score -24.157 -1.12512 12 12 Pose