FAIRMol

Reverse docking explorer

Search one compound across many targets or scan the strongest compound-target pairs in the active database. The combined reverse-docking score uses a normalized docking-score estimator together with an interaction-fingerprint component.

DB SELECTIONExplorer results are being read from this database.
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2 compounds in matrix 5 best compound-target hits listed 5 targets
• Combined reverse-docking score = 65% normalized docking-score estimator + 35% interaction-fingerprint component.
• When a native ligand exists for an experiment, the interaction-fingerprint component is driven by similarity to the native contact/H-bond pattern.
• When no native ligand exists, the interaction-fingerprint component falls back to contact richness within the experiment (normalized contacts and H-bonds).

Compounds × targets matrix

Each cell shows the best combined reverse-docking score found for that compound on that target. Blank cells mean no imported pose passed the current filters.
Compound Best Mean Targets T01T02T16T17T18
TC354
[H]N(CCc1ccc([N+]([H])([H])[H])cc1)C1=C(/C=C/C2=[N+](C)c3ccccc3C2(C)C)CCC/C1=C\C=C1\N(C)c2ccccc2C1(C)C
0.827 0.794 4 0.81 0.83 0.76 0.79
TC354
[H]N(CCc1ccc(N([H])[H])cc1)C1=C(/C=C/C2=[N+](C)c3ccccc3C2(C)C)CCC/C1=C\C=C1\N(C)c2ccccc2C1(C)C
0.816 0.816 1 0.82

Best compound-target hits

The score column is the combined reverse-docking score. The next two columns expose its components: normalized score-estimator and interaction fingerprint.
CompoundTargetExperimentCombinedScore partIFP partIFP modeMetricDock scoreInter normContactsHB
TC354
[H]N(CCc1ccc([N+]([H])([H])[H])cc1)C1=C(/C=C/C2=[N+](C)c3ccccc3C2(C)C)CCC/C1=C\C=C1\N(C)c2ccccc2C1(C)C
T02
native IFP available
T02
selection_import_t02
0.827 1.000 0.507 native_similarity final_rank_score -22.3914 -0.579766 18 2 Pose
TC354
[H]N(CCc1ccc(N([H])[H])cc1)C1=C(/C=C/C2=[N+](C)c3ccccc3C2(C)C)CCC/C1=C\C=C1\N(C)c2ccccc2C1(C)C
T17
native IFP available
T17
selection_import_t17
0.816 1.000 0.475 native_similarity final_rank_score -17.7761 -0.518156 21 3 Pose
TC354
[H]N(CCc1ccc([N+]([H])([H])[H])cc1)C1=C(/C=C/C2=[N+](C)c3ccccc3C2(C)C)CCC/C1=C\C=C1\N(C)c2ccccc2C1(C)C
T01
native IFP available
T01
selection_import_t01
0.805 1.000 0.443 native_similarity final_rank_score -23.0597 -0.634928 16 2 Pose
TC354
[H]N(CCc1ccc([N+]([H])([H])[H])cc1)C1=C(/C=C/C2=[N+](C)c3ccccc3C2(C)C)CCC/C1=C\C=C1\N(C)c2ccccc2C1(C)C
T18
native IFP available
T18
selection_import_t18
0.786 1.000 0.388 native_similarity final_rank_score -16.6641 -0.475706 16 3 Pose
TC354
[H]N(CCc1ccc([N+]([H])([H])[H])cc1)C1=C(/C=C/C2=[N+](C)c3ccccc3C2(C)C)CCC/C1=C\C=C1\N(C)c2ccccc2C1(C)C
T16
native IFP available
T16
selection_import_t16
0.756 1.000 0.302 native_similarity final_rank_score -22.034 -0.539598 17 3 Pose