FAIRMol

Reverse docking explorer

Search one compound across many targets or scan the strongest compound-target pairs in the active database. The combined reverse-docking score uses a normalized docking-score estimator together with an interaction-fingerprint component.

DB SELECTIONExplorer results are being read from this database.
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2 compounds in matrix 3 best compound-target hits listed 3 targets
• Combined reverse-docking score = 65% normalized docking-score estimator + 35% interaction-fingerprint component.
• When a native ligand exists for an experiment, the interaction-fingerprint component is driven by similarity to the native contact/H-bond pattern.
• When no native ligand exists, the interaction-fingerprint component falls back to contact richness within the experiment (normalized contacts and H-bonds).

Compounds × targets matrix

Each cell shows the best combined reverse-docking score found for that compound on that target. Blank cells mean no imported pose passed the current filters.
Compound Best Mean Targets T01T15T16
OSA_Lib_52
[H][N+]([H])([H])[C@@H]1C[C@]2([N+]3([H])CCCCC3)C[C@H](c3ccccc3)[C@H]1[C@@H](c1ccccc1)C2
0.860 0.826 2 0.86 0.79
OSA_Lib_52
[H][N+]([H])([H])[C@H]1C[C@]2(N3CCCCC3)C[C@H](c3ccccc3)[C@H]1[C@H](c1ccccc1)C2
0.763 0.763 1 0.76

Best compound-target hits

The score column is the combined reverse-docking score. The next two columns expose its components: normalized score-estimator and interaction fingerprint.
CompoundTargetExperimentCombinedScore partIFP partIFP modeMetricDock scoreInter normContactsHB
OSA_Lib_52
[H][N+]([H])([H])[C@@H]1C[C@]2([N+]3([H])CCCCC3)C[C@H](c3ccccc3)[C@H]1[C@@H](c1ccccc1)C2
T01
native IFP available
T01
selection_import_t01
0.860 1.000 0.600 native_similarity final_rank_score -25.7271 -1.00743 18 2 Pose
OSA_Lib_52
[H][N+]([H])([H])[C@@H]1C[C@]2([N+]3([H])CCCCC3)C[C@H](c3ccccc3)[C@H]1[C@@H](c1ccccc1)C2
T15
native IFP available
T15
selection_import_t15
0.793 1.000 0.408 native_similarity final_rank_score -25.1895 -0.928802 14 3 Pose
OSA_Lib_52
[H][N+]([H])([H])[C@H]1C[C@]2(N3CCCCC3)C[C@H](c3ccccc3)[C@H]1[C@H](c1ccccc1)C2
T16
native IFP available
T16
selection_import_t16
0.763 1.000 0.322 native_similarity final_rank_score -24.9996 -0.959833 14 4 Pose