FAIRMol

Reverse docking explorer

Search one compound across many targets or scan the strongest compound-target pairs in the active database. The combined reverse-docking score uses a normalized docking-score estimator together with an interaction-fingerprint component.

DB SELECTIONExplorer results are being read from this database.
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2 compounds in matrix 5 best compound-target hits listed 5 targets
• Combined reverse-docking score = 65% normalized docking-score estimator + 35% interaction-fingerprint component.
• When a native ligand exists for an experiment, the interaction-fingerprint component is driven by similarity to the native contact/H-bond pattern.
• When no native ligand exists, the interaction-fingerprint component falls back to contact richness within the experiment (normalized contacts and H-bonds).

Compounds × targets matrix

Each cell shows the best combined reverse-docking score found for that compound on that target. Blank cells mean no imported pose passed the current filters.
Compound Best Mean Targets T01T03T15T16T18
OSA_Lib_306
[H][N@+]1(Cc2cccnc2)C[C@H]2[C@@H](c3ccccc3)C[C@](N3CCCC3)(C[C@@H]2c2ccccc2)C1
0.864 0.819 4 0.84 0.86 0.81 0.76
OSA_Lib_306
[H][N@+]1(Cc2cccnc2)C[C@@H]2[C@@H](c3ccccc3)C[C@@](N3CCCC3)(C[C@H]2c2ccccc2)C1
0.777 0.777 1 0.78

Best compound-target hits

The score column is the combined reverse-docking score. The next two columns expose its components: normalized score-estimator and interaction fingerprint.
CompoundTargetExperimentCombinedScore partIFP partIFP modeMetricDock scoreInter normContactsHB
OSA_Lib_306
[H][N@+]1(Cc2cccnc2)C[C@H]2[C@@H](c3ccccc3)C[C@](N3CCCC3)(C[C@@H]2c2ccccc2)C1
T03
native IFP available
T03
selection_import_t03
0.864 1.000 0.611 native_similarity final_rank_score -24.7326 -0.813951 20 2 Pose
OSA_Lib_306
[H][N@+]1(Cc2cccnc2)C[C@H]2[C@@H](c3ccccc3)C[C@](N3CCCC3)(C[C@@H]2c2ccccc2)C1
T01
native IFP available
T01
selection_import_t01
0.844 1.000 0.555 native_similarity final_rank_score -25.0702 -0.772726 19 1 Pose
OSA_Lib_306
[H][N@+]1(Cc2cccnc2)C[C@H]2[C@@H](c3ccccc3)C[C@](N3CCCC3)(C[C@@H]2c2ccccc2)C1
T15
native IFP available
T15
selection_import_t15
0.809 1.000 0.453 native_similarity final_rank_score -24.3593 -0.739339 15 1 Pose
OSA_Lib_306
[H][N@+]1(Cc2cccnc2)C[C@@H]2[C@@H](c3ccccc3)C[C@@](N3CCCC3)(C[C@H]2c2ccccc2)C1
T18
native IFP available
T18
selection_import_t18
0.777 1.000 0.362 native_similarity final_rank_score -19.2691 -0.638909 13 2 Pose
OSA_Lib_306
[H][N@+]1(Cc2cccnc2)C[C@H]2[C@@H](c3ccccc3)C[C@](N3CCCC3)(C[C@@H]2c2ccccc2)C1
T16
native IFP available
T16
selection_import_t16
0.760 1.000 0.315 native_similarity final_rank_score -22.9119 -0.703428 15 2 Pose