FAIRMol

Reverse docking explorer

Search one compound across many targets or scan the strongest compound-target pairs in the active database. The combined reverse-docking score uses a normalized docking-score estimator together with an interaction-fingerprint component.

DB SELECTIONExplorer results are being read from this database.
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2 compounds in matrix 13 best compound-target hits listed 13 targets
• Combined reverse-docking score = 65% normalized docking-score estimator + 35% interaction-fingerprint component.
• When a native ligand exists for an experiment, the interaction-fingerprint component is driven by similarity to the native contact/H-bond pattern.
• When no native ligand exists, the interaction-fingerprint component falls back to contact richness within the experiment (normalized contacts and H-bonds).

Compounds × targets matrix

Each cell shows the best combined reverse-docking score found for that compound on that target. Blank cells mean no imported pose passed the current filters.
Compound Best Mean Targets T01T02T03T07T08T10T12T13T14T15T16T18T21
OHD_MAC_16
[H]OCCCOc1cccc(N([H])c2c3ncn([H])/c(=N\[N+]([H])=C\c4ccc(O[H])c(O[H])c4)c3nc[n+]2[H])c1
0.947 0.842 10 0.82 0.82 0.77 0.87 0.84 0.95 0.94 0.87 0.76 0.78
OHD_MAC_16
[H]OCCCOc1cccc(N([H])c2ncnc3c(N([H])/N=C/c4ccc(O[H])c(O[H])c4)ncnc23)c1
0.945 0.868 3 0.85 0.80 0.94

Best compound-target hits

The score column is the combined reverse-docking score. The next two columns expose its components: normalized score-estimator and interaction fingerprint.
CompoundTargetExperimentCombinedScore partIFP partIFP modeMetricDock scoreInter normContactsHB
OHD_MAC_16
[H]OCCCOc1cccc(N([H])c2c3ncn([H])/c(=N\[N+]([H])=C\c4ccc(O[H])c(O[H])c4)c3nc[n+]2[H])c1
T10
native IFP available
T10
selection_import_t10
0.947 1.000 0.849 native_similarity final_rank_score -25.8714 -1.00391 20 11 Pose
OHD_MAC_16
[H]OCCCOc1cccc(N([H])c2ncnc3c(N([H])/N=C/c4ccc(O[H])c(O[H])c4)ncnc23)c1
T21
native IFP available
T21
selection_import_t21
0.945 1.000 0.842 native_similarity final_rank_score -22.5587 -0.795842 18 14 Pose
OHD_MAC_16
[H]OCCCOc1cccc(N([H])c2c3ncn([H])/c(=N\[N+]([H])=C\c4ccc(O[H])c(O[H])c4)c3nc[n+]2[H])c1
T12
native IFP available
T12
selection_import_t12
0.936 1.000 0.817 native_similarity final_rank_score -33.5625 -1.0808 19 15 Pose
OHD_MAC_16
[H]OCCCOc1cccc(N([H])c2c3ncn([H])/c(=N\[N+]([H])=C\c4ccc(O[H])c(O[H])c4)c3nc[n+]2[H])c1
T07
native IFP available
T07
selection_import_t07
0.869 1.000 0.627 native_similarity final_rank_score -20.5158 -1.00748 20 10 Pose
OHD_MAC_16
[H]OCCCOc1cccc(N([H])c2c3ncn([H])/c(=N\[N+]([H])=C\c4ccc(O[H])c(O[H])c4)c3nc[n+]2[H])c1
T13
native IFP available
T13
selection_import_t13
0.865 1.000 0.615 native_similarity final_rank_score -25.4105 -0.952554 20 11 Pose
OHD_MAC_16
[H]OCCCOc1cccc(N([H])c2ncnc3c(N([H])/N=C/c4ccc(O[H])c(O[H])c4)ncnc23)c1
T16
native IFP available
T16
selection_import_t16
0.854 1.000 0.582 native_similarity final_rank_score -20.4372 -0.780129 17 5 Pose
OHD_MAC_16
[H]OCCCOc1cccc(N([H])c2c3ncn([H])/c(=N\[N+]([H])=C\c4ccc(O[H])c(O[H])c4)c3nc[n+]2[H])c1
T08
native IFP available
T08
selection_import_t08
0.842 1.000 0.550 native_similarity final_rank_score -31.5208 -1.28243 17 10 Pose
OHD_MAC_16
[H]OCCCOc1cccc(N([H])c2c3ncn([H])/c(=N\[N+]([H])=C\c4ccc(O[H])c(O[H])c4)c3nc[n+]2[H])c1
T01
native IFP available
T01
selection_import_t01
0.819 1.000 0.484 native_similarity final_rank_score -25.5705 -0.863295 18 6 Pose
OHD_MAC_16
[H]OCCCOc1cccc(N([H])c2c3ncn([H])/c(=N\[N+]([H])=C\c4ccc(O[H])c(O[H])c4)c3nc[n+]2[H])c1
T02
native IFP available
T02
selection_import_t02
0.819 1.000 0.484 native_similarity final_rank_score -23.7773 -0.84998 18 6 Pose
OHD_MAC_16
[H]OCCCOc1cccc(N([H])c2ncnc3c(N([H])/N=C/c4ccc(O[H])c(O[H])c4)ncnc23)c1
T18
native IFP available
T18
selection_import_t18
0.804 1.000 0.441 native_similarity final_rank_score -20.8359 -0.74205 16 6 Pose
OHD_MAC_16
[H]OCCCOc1cccc(N([H])c2c3ncn([H])/c(=N\[N+]([H])=C\c4ccc(O[H])c(O[H])c4)c3nc[n+]2[H])c1
T15
native IFP available
T15
selection_import_t15
0.783 1.000 0.379 native_similarity final_rank_score -20.8598 -0.706094 17 5 Pose
OHD_MAC_16
[H]OCCCOc1cccc(N([H])c2c3ncn([H])/c(=N\[N+]([H])=C\c4ccc(O[H])c(O[H])c4)c3nc[n+]2[H])c1
T03
native IFP available
T03
selection_import_t03
0.775 1.000 0.356 native_similarity final_rank_score -21.6169 -0.824084 14 6 Pose
OHD_MAC_16
[H]OCCCOc1cccc(N([H])c2c3ncn([H])/c(=N\[N+]([H])=C\c4ccc(O[H])c(O[H])c4)c3nc[n+]2[H])c1
T14
native IFP available
T14
selection_import_t14
0.765 1.000 0.327 native_similarity final_rank_score -21.9396 -0.766228 14 10 Pose