FAIRMol

Reverse docking explorer

Search one compound across many targets or scan the strongest compound-target pairs in the active database. The combined reverse-docking score uses a normalized docking-score estimator together with an interaction-fingerprint component.

DB SELECTIONExplorer results are being read from this database.
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2 compounds in matrix 5 best compound-target hits listed 5 targets
• Combined reverse-docking score = 65% normalized docking-score estimator + 35% interaction-fingerprint component.
• When a native ligand exists for an experiment, the interaction-fingerprint component is driven by similarity to the native contact/H-bond pattern.
• When no native ligand exists, the interaction-fingerprint component falls back to contact richness within the experiment (normalized contacts and H-bonds).

Compounds × targets matrix

Each cell shows the best combined reverse-docking score found for that compound on that target. Blank cells mean no imported pose passed the current filters.
Compound Best Mean Targets T01T02T08T09T14
OHD_ACDS_33
[H]n1cc(C(C[N+]([H])([H])Cc2ccc(F)cc2)c2cn([H])c3cc(Br)ccc23)c2ccc(Br)cc21
0.916 0.851 2 0.92 0.79
OHD_ACDS_33
[H]N(Cc1ccc(F)cc1)CC(c1cn([H])c2cc(Br)ccc12)c1cn([H])c2cc(Br)ccc12
0.893 0.872 3 0.89 0.85 0.87

Best compound-target hits

The score column is the combined reverse-docking score. The next two columns expose its components: normalized score-estimator and interaction fingerprint.
CompoundTargetExperimentCombinedScore partIFP partIFP modeMetricDock scoreInter normContactsHB
OHD_ACDS_33
[H]n1cc(C(C[N+]([H])([H])Cc2ccc(F)cc2)c2cn([H])c3cc(Br)ccc23)c2ccc(Br)cc21
T02
native IFP available
T02
selection_import_t02
0.916 1.000 0.760 native_similarity final_rank_score -25.018 -0.880069 21 2 Pose
OHD_ACDS_33
[H]N(Cc1ccc(F)cc1)CC(c1cn([H])c2cc(Br)ccc12)c1cn([H])c2cc(Br)ccc12
T01
native IFP available
T01
selection_import_t01
0.893 1.000 0.693 native_similarity final_rank_score -26.0602 -0.843549 19 2 Pose
OHD_ACDS_33
[H]N(Cc1ccc(F)cc1)CC(c1cn([H])c2cc(Br)ccc12)c1cn([H])c2cc(Br)ccc12
T09
native IFP available
T09
selection_import_t09
0.872 1.000 0.634 native_similarity final_rank_score -25.406 -0.917305 19 2 Pose
OHD_ACDS_33
[H]N(Cc1ccc(F)cc1)CC(c1cn([H])c2cc(Br)ccc12)c1cn([H])c2cc(Br)ccc12
T08
native IFP available
T08
selection_import_t08
0.851 1.000 0.574 native_similarity final_rank_score -34.2668 -1.12814 19 2 Pose
OHD_ACDS_33
[H]n1cc(C(C[N+]([H])([H])Cc2ccc(F)cc2)c2cn([H])c3cc(Br)ccc23)c2ccc(Br)cc21
T14
native IFP available
T14
selection_import_t14
0.786 1.000 0.388 native_similarity final_rank_score -18.7206 -0.773857 12 3 Pose