FAIRMol

Reverse docking explorer

Search one compound across many targets or scan the strongest compound-target pairs in the active database. The combined reverse-docking score uses a normalized docking-score estimator together with an interaction-fingerprint component.

DB SELECTIONExplorer results are being read from this database.
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2 compounds in matrix 9 best compound-target hits listed 9 targets
• Combined reverse-docking score = 65% normalized docking-score estimator + 35% interaction-fingerprint component.
• When a native ligand exists for an experiment, the interaction-fingerprint component is driven by similarity to the native contact/H-bond pattern.
• When no native ligand exists, the interaction-fingerprint component falls back to contact richness within the experiment (normalized contacts and H-bonds).

Compounds × targets matrix

Each cell shows the best combined reverse-docking score found for that compound on that target. Blank cells mean no imported pose passed the current filters.
Compound Best Mean Targets T01T02T04T06T07T08T11T16T20
NMT-TY0562
[H]N([H])c1nc(N([H])[H])[n+]([H])cc1NS(=O)(=O)c1ccc(N([H])C(C)=O)cc1
0.919 0.840 5 0.80 0.80 0.92 0.90 0.78
NMT-TY0562
[H]N([H])c1ncc(NS(=O)(=O)c2ccc(N([H])C(C)=O)cc2)c(N([H])[H])n1
0.902 0.853 4 0.90 0.89 0.75 0.87

Best compound-target hits

The score column is the combined reverse-docking score. The next two columns expose its components: normalized score-estimator and interaction fingerprint.
CompoundTargetExperimentCombinedScore partIFP partIFP modeMetricDock scoreInter normContactsHB
NMT-TY0562
[H]N([H])c1nc(N([H])[H])[n+]([H])cc1NS(=O)(=O)c1ccc(N([H])C(C)=O)cc1
T07
native IFP available
T07
selection_import_t07
0.919 1.000 0.769 native_similarity final_rank_score -30.1885 -1.49349 16 10 Pose
NMT-TY0562
[H]N([H])c1ncc(NS(=O)(=O)c2ccc(N([H])C(C)=O)cc2)c(N([H])[H])n1
T04
native IFP available
T04
selection_import_t04
0.902 1.000 0.719 native_similarity final_rank_score -25.3727 -1.24137 13 6 Pose
NMT-TY0562
[H]N([H])c1nc(N([H])[H])[n+]([H])cc1NS(=O)(=O)c1ccc(N([H])C(C)=O)cc1
T08
native IFP available
T08
selection_import_t08
0.901 1.000 0.717 native_similarity final_rank_score -29.9963 -1.46166 16 9 Pose
NMT-TY0562
[H]N([H])c1ncc(NS(=O)(=O)c2ccc(N([H])C(C)=O)cc2)c(N([H])[H])n1
T06
native IFP available
T06
selection_import_t06
0.887 1.000 0.676 native_similarity final_rank_score -18.1033 -1.05343 20 8 Pose
NMT-TY0562
[H]N([H])c1ncc(NS(=O)(=O)c2ccc(N([H])C(C)=O)cc2)c(N([H])[H])n1
T20
native IFP available
T20
selection_import_t20
0.874 1.000 0.641 native_similarity final_rank_score -19.7272 -0.948695 10 6 Pose
NMT-TY0562
[H]N([H])c1nc(N([H])[H])[n+]([H])cc1NS(=O)(=O)c1ccc(N([H])C(C)=O)cc1
T01
native IFP available
T01
selection_import_t01
0.800 1.000 0.429 native_similarity final_rank_score -23.3606 -1.18394 19 11 Pose
NMT-TY0562
[H]N([H])c1nc(N([H])[H])[n+]([H])cc1NS(=O)(=O)c1ccc(N([H])C(C)=O)cc1
T02
native IFP available
T02
selection_import_t02
0.800 1.000 0.429 native_similarity final_rank_score -23.1368 -1.19357 19 11 Pose
NMT-TY0562
[H]N([H])c1nc(N([H])[H])[n+]([H])cc1NS(=O)(=O)c1ccc(N([H])C(C)=O)cc1
T11
native IFP available
T11
selection_import_t11
0.778 1.000 0.365 native_similarity final_rank_score -22.8829 -1.1435 15 7 Pose
NMT-TY0562
[H]N([H])c1ncc(NS(=O)(=O)c2ccc(N([H])C(C)=O)cc2)c(N([H])[H])n1
T16
native IFP available
T16
selection_import_t16
0.749 1.000 0.283 native_similarity final_rank_score -22.7772 -1.0463 12 9 Pose