FAIRMol

Reverse docking explorer

Search one compound across many targets or scan the strongest compound-target pairs in the active database. The combined reverse-docking score uses a normalized docking-score estimator together with an interaction-fingerprint component.

DB SELECTIONExplorer results are being read from this database.
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1 compounds in matrix 14 best compound-target hits listed 14 targets
• Combined reverse-docking score = 65% normalized docking-score estimator + 35% interaction-fingerprint component.
• When a native ligand exists for an experiment, the interaction-fingerprint component is driven by similarity to the native contact/H-bond pattern.
• When no native ligand exists, the interaction-fingerprint component falls back to contact richness within the experiment (normalized contacts and H-bonds).

Compounds × targets matrix

Each cell shows the best combined reverse-docking score found for that compound on that target. Blank cells mean no imported pose passed the current filters.
Compound Best Mean Targets T01T04T05T06T07T08T09T10T11T12T14T16T19T22
NMT-TY0549
[H]N([H])c1nc(N([H])[H])n([H])c(=O)c1N([H])C/C(O)=N/S(=O)(=O)c1ccc(N([H])C(C)=O)cc1
0.960 0.879 14 0.92 0.93 0.89 0.93 0.91 0.90 0.79 0.92 0.91 0.96 0.79 0.81 0.77 0.87

Best compound-target hits

The score column is the combined reverse-docking score. The next two columns expose its components: normalized score-estimator and interaction fingerprint.
CompoundTargetExperimentCombinedScore partIFP partIFP modeMetricDock scoreInter normContactsHB
NMT-TY0549
[H]N([H])c1nc(N([H])[H])n([H])c(=O)c1N([H])C/C(O)=N/S(=O)(=O)c1ccc(N([H])C(C)=O)cc1
T12
native IFP available
T12
selection_import_t12
0.960 1.000 0.886 native_similarity final_rank_score -36.0618 -1.2862 17 15 Pose
NMT-TY0549
[H]N([H])c1nc(N([H])[H])n([H])c(=O)c1N([H])C/C(O)=N/S(=O)(=O)c1ccc(N([H])C(C)=O)cc1
T06
native IFP available
T06
selection_import_t06
0.931 1.000 0.802 native_similarity final_rank_score -22.8583 -0.887788 18 6 Pose
NMT-TY0549
[H]N([H])c1nc(N([H])[H])n([H])c(=O)c1N([H])C/C(O)=N/S(=O)(=O)c1ccc(N([H])C(C)=O)cc1
T04
native IFP available
T04
selection_import_t04
0.927 1.000 0.793 native_similarity final_rank_score -24.9818 -0.911074 15 7 Pose
NMT-TY0549
[H]N([H])c1nc(N([H])[H])n([H])c(=O)c1N([H])C/C(O)=N/S(=O)(=O)c1ccc(N([H])C(C)=O)cc1
T01
native IFP available
T01
selection_import_t01
0.922 1.000 0.779 native_similarity final_rank_score -22.8123 -0.963314 19 12 Pose
NMT-TY0549
[H]N([H])c1nc(N([H])[H])n([H])c(=O)c1N([H])C/C(O)=N/S(=O)(=O)c1ccc(N([H])C(C)=O)cc1
T10
native IFP available
T10
selection_import_t10
0.920 1.000 0.771 native_similarity final_rank_score -29.1414 -1.00534 16 16 Pose
NMT-TY0549
[H]N([H])c1nc(N([H])[H])n([H])c(=O)c1N([H])C/C(O)=N/S(=O)(=O)c1ccc(N([H])C(C)=O)cc1
T07
native IFP available
T07
selection_import_t07
0.911 1.000 0.745 native_similarity final_rank_score -32.8271 -1.25212 20 13 Pose
NMT-TY0549
[H]N([H])c1nc(N([H])[H])n([H])c(=O)c1N([H])C/C(O)=N/S(=O)(=O)c1ccc(N([H])C(C)=O)cc1
T11
native IFP available
T11
selection_import_t11
0.908 1.000 0.737 native_similarity final_rank_score -30.1625 -1.06372 15 10 Pose
NMT-TY0549
[H]N([H])c1nc(N([H])[H])n([H])c(=O)c1N([H])C/C(O)=N/S(=O)(=O)c1ccc(N([H])C(C)=O)cc1
T08
native IFP available
T08
selection_import_t08
0.901 1.000 0.717 native_similarity final_rank_score -34.4996 -1.23884 21 16 Pose
NMT-TY0549
[H]N([H])c1nc(N([H])[H])n([H])c(=O)c1N([H])C/C(O)=N/S(=O)(=O)c1ccc(N([H])C(C)=O)cc1
T05
native IFP available
T05
selection_import_t05
0.886 1.000 0.674 native_similarity final_rank_score -36.2843 -1.31147 18 14 Pose
NMT-TY0549
[H]N([H])c1nc(N([H])[H])n([H])c(=O)c1N([H])C/C(O)=N/S(=O)(=O)c1ccc(N([H])C(C)=O)cc1
T22
native IFP available
T22
selection_import_t22
0.875 1.000 0.642 native_similarity final_rank_score -31.3287 -1.2144 26 15 Pose
NMT-TY0549
[H]N([H])c1nc(N([H])[H])n([H])c(=O)c1N([H])C/C(O)=N/S(=O)(=O)c1ccc(N([H])C(C)=O)cc1
T16
native IFP available
T16
selection_import_t16
0.807 1.000 0.450 native_similarity final_rank_score -26.0956 -0.898096 13 7 Pose
NMT-TY0549
[H]N([H])c1nc(N([H])[H])n([H])c(=O)c1N([H])C/C(O)=N/S(=O)(=O)c1ccc(N([H])C(C)=O)cc1
T14
native IFP available
T14
selection_import_t14
0.793 1.000 0.409 native_similarity final_rank_score -26.3877 -0.915736 13 13 Pose
NMT-TY0549
[H]N([H])c1nc(N([H])[H])n([H])c(=O)c1N([H])C/C(O)=N/S(=O)(=O)c1ccc(N([H])C(C)=O)cc1
T09
native IFP available
T09
selection_import_t09
0.788 1.000 0.394 native_similarity final_rank_score -26.3261 -1.07778 17 11 Pose
NMT-TY0549
[H]N([H])c1nc(N([H])[H])n([H])c(=O)c1N([H])C/C(O)=N/S(=O)(=O)c1ccc(N([H])C(C)=O)cc1
T19
native IFP available
T19
selection_import_t19
0.774 1.000 0.354 native_similarity final_rank_score -32.7493 -1.21946 15 11 Pose