FAIRMol

Reverse docking explorer

Search one compound across many targets or scan the strongest compound-target pairs in the active database. The combined reverse-docking score uses a normalized docking-score estimator together with an interaction-fingerprint component.

DB SELECTIONExplorer results are being read from this database.
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2 compounds in matrix 4 best compound-target hits listed 4 targets
• Combined reverse-docking score = 65% normalized docking-score estimator + 35% interaction-fingerprint component.
• When a native ligand exists for an experiment, the interaction-fingerprint component is driven by similarity to the native contact/H-bond pattern.
• When no native ligand exists, the interaction-fingerprint component falls back to contact richness within the experiment (normalized contacts and H-bonds).

Compounds × targets matrix

Each cell shows the best combined reverse-docking score found for that compound on that target. Blank cells mean no imported pose passed the current filters.
Compound Best Mean Targets T01T10T11T20
MK33
[H]Oc1c(C)c(C)c2c(c1CC[N@+]([H])(C)CCc1ccc(NS(C)(=O)=O)cc1)CCC(C)(C)O2
0.962 0.881 3 0.84 0.84 0.96
MK33
[H]Oc1c(C)c(C)c2c(c1CCN(C)CCc1ccc(N([H])S(C)(=O)=O)cc1)CCC(C)(C)O2
0.933 0.933 1 0.93

Best compound-target hits

The score column is the combined reverse-docking score. The next two columns expose its components: normalized score-estimator and interaction fingerprint.
CompoundTargetExperimentCombinedScore partIFP partIFP modeMetricDock scoreInter normContactsHB
MK33
[H]Oc1c(C)c(C)c2c(c1CC[N@+]([H])(C)CCc1ccc(NS(C)(=O)=O)cc1)CCC(C)(C)O2
T20
native IFP available
T20
selection_import_t20
0.962 1.000 0.891 native_similarity final_rank_score -16.2823 -0.604967 11 8 Pose
MK33
[H]Oc1c(C)c(C)c2c(c1CCN(C)CCc1ccc(N([H])S(C)(=O)=O)cc1)CCC(C)(C)O2
T10
native IFP available
T10
selection_import_t10
0.933 1.000 0.809 native_similarity final_rank_score -23.9872 -0.790534 15 11 Pose
MK33
[H]Oc1c(C)c(C)c2c(c1CC[N@+]([H])(C)CCc1ccc(NS(C)(=O)=O)cc1)CCC(C)(C)O2
T01
native IFP available
T01
selection_import_t01
0.840 1.000 0.544 native_similarity final_rank_score -22.2376 -0.843483 18 3 Pose
MK33
[H]Oc1c(C)c(C)c2c(c1CC[N@+]([H])(C)CCc1ccc(NS(C)(=O)=O)cc1)CCC(C)(C)O2
T11
native IFP available
T11
selection_import_t11
0.840 1.000 0.543 native_similarity final_rank_score -17.9078 -0.830247 17 4 Pose