FAIRMol

Reverse docking explorer

Search one compound across many targets or scan the strongest compound-target pairs in the active database. The combined reverse-docking score uses a normalized docking-score estimator together with an interaction-fingerprint component.

DB SELECTIONExplorer results are being read from this database.
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4 compounds in matrix 4 best compound-target hits listed 4 targets
• Combined reverse-docking score = 65% normalized docking-score estimator + 35% interaction-fingerprint component.
• When a native ligand exists for an experiment, the interaction-fingerprint component is driven by similarity to the native contact/H-bond pattern.
• When no native ligand exists, the interaction-fingerprint component falls back to contact richness within the experiment (normalized contacts and H-bonds).

Compounds × targets matrix

Each cell shows the best combined reverse-docking score found for that compound on that target. Blank cells mean no imported pose passed the current filters.
Compound Best Mean Targets T05T14T20T21
MK132
[H]O[C@@H]1[C@H](O[H])[C@@H](CO[N+](=O)O)O[C@@H]1n1cnc2c(N([H])Cc3ccccc3)ncnc21
0.963 0.963 1 0.96
MK132
[H]O[C@@H]1[C@H](O[H])[C@H](CO[N+](=O)O)O[C@H]1n1cnc2c(N([H])Cc3ccccc3)ncnc21
0.850 0.850 1 0.85
MK132
[H]O[C@@H]1[C@@H](O[H])[C@@H](CO[N+](=O)O)O[C@H]1n1cnc2c(N([H])Cc3ccccc3)ncnc21
0.824 0.824 1 0.82
MK132
[H]O[C@@H]1[C@H](O[H])[C@@H](CO[N+](=O)O)O[C@H]1n1cnc2c(N([H])Cc3ccccc3)ncnc21
0.822 0.822 1 0.82

Best compound-target hits

The score column is the combined reverse-docking score. The next two columns expose its components: normalized score-estimator and interaction fingerprint.
CompoundTargetExperimentCombinedScore partIFP partIFP modeMetricDock scoreInter normContactsHB
MK132
[H]O[C@@H]1[C@H](O[H])[C@@H](CO[N+](=O)O)O[C@@H]1n1cnc2c(N([H])Cc3ccccc3)ncnc21
T21
native IFP available
T21
selection_import_t21
0.963 1.000 0.893 native_similarity final_rank_score -24.4043 -0.86354 16 16 Pose
MK132
[H]O[C@@H]1[C@H](O[H])[C@H](CO[N+](=O)O)O[C@H]1n1cnc2c(N([H])Cc3ccccc3)ncnc21
T05
native IFP available
T05
selection_import_t05
0.850 1.000 0.572 native_similarity final_rank_score -31.3065 -1.0204 19 11 Pose
MK132
[H]O[C@@H]1[C@@H](O[H])[C@@H](CO[N+](=O)O)O[C@H]1n1cnc2c(N([H])Cc3ccccc3)ncnc21
T20
native IFP available
T20
selection_import_t20
0.824 1.000 0.496 native_similarity final_rank_score -19.3375 -0.654802 11 7 Pose
MK132
[H]O[C@@H]1[C@H](O[H])[C@@H](CO[N+](=O)O)O[C@H]1n1cnc2c(N([H])Cc3ccccc3)ncnc21
T14
native IFP available
T14
selection_import_t14
0.822 1.000 0.491 native_similarity final_rank_score -24.7009 -0.807174 15 12 Pose