FAIRMol

Reverse docking explorer

Search one compound across many targets or scan the strongest compound-target pairs in the active database. The combined reverse-docking score uses a normalized docking-score estimator together with an interaction-fingerprint component.

DB SELECTIONExplorer results are being read from this database.
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2 compounds in matrix 6 best compound-target hits listed 6 targets
• Combined reverse-docking score = 65% normalized docking-score estimator + 35% interaction-fingerprint component.
• When a native ligand exists for an experiment, the interaction-fingerprint component is driven by similarity to the native contact/H-bond pattern.
• When no native ligand exists, the interaction-fingerprint component falls back to contact richness within the experiment (normalized contacts and H-bonds).

Compounds × targets matrix

Each cell shows the best combined reverse-docking score found for that compound on that target. Blank cells mean no imported pose passed the current filters.
Compound Best Mean Targets T01T10T11T13T17T21
MK10
[H]Oc1c(C)c(C)c2c(c1CN1CCN(c3ccc(N([H])S(C)(=O)=O)cc3)CC1)CCC(C)(C)O2
0.933 0.897 3 0.93 0.83 0.93
MK10
[H]Oc1c(C)c(C)c2c(c1C[N+]1([H])CCN(c3ccc(N([H])S(C)(=O)=O)cc3)CC1)CCC(C)(C)O2
0.893 0.873 3 0.87 0.89 0.86

Best compound-target hits

The score column is the combined reverse-docking score. The next two columns expose its components: normalized score-estimator and interaction fingerprint.
CompoundTargetExperimentCombinedScore partIFP partIFP modeMetricDock scoreInter normContactsHB
MK10
[H]Oc1c(C)c(C)c2c(c1CN1CCN(c3ccc(N([H])S(C)(=O)=O)cc3)CC1)CCC(C)(C)O2
T10
native IFP available
T10
selection_import_t10
0.933 1.000 0.809 native_similarity final_rank_score -23.921 -0.752691 15 10 Pose
MK10
[H]Oc1c(C)c(C)c2c(c1CN1CCN(c3ccc(N([H])S(C)(=O)=O)cc3)CC1)CCC(C)(C)O2
T21
native IFP available
T21
selection_import_t21
0.929 1.000 0.798 native_similarity final_rank_score -23.2356 -0.75256 17 14 Pose
MK10
[H]Oc1c(C)c(C)c2c(c1C[N+]1([H])CCN(c3ccc(N([H])S(C)(=O)=O)cc3)CC1)CCC(C)(C)O2
T13
native IFP available
T13
selection_import_t13
0.893 1.000 0.694 native_similarity final_rank_score -23.8486 -0.856708 17 7 Pose
MK10
[H]Oc1c(C)c(C)c2c(c1C[N+]1([H])CCN(c3ccc(N([H])S(C)(=O)=O)cc3)CC1)CCC(C)(C)O2
T01
native IFP available
T01
selection_import_t01
0.871 1.000 0.630 native_similarity final_rank_score -26.4227 -0.7986 20 2 Pose
MK10
[H]Oc1c(C)c(C)c2c(c1C[N+]1([H])CCN(c3ccc(N([H])S(C)(=O)=O)cc3)CC1)CCC(C)(C)O2
T17
native IFP available
T17
selection_import_t17
0.855 1.000 0.587 native_similarity final_rank_score -25.8817 -0.768814 20 6 Pose
MK10
[H]Oc1c(C)c(C)c2c(c1CN1CCN(c3ccc(N([H])S(C)(=O)=O)cc3)CC1)CCC(C)(C)O2
T11
native IFP available
T11
selection_import_t11
0.827 1.000 0.507 native_similarity final_rank_score -22.6819 -0.810619 21 2 Pose