FAIRMol

Reverse docking explorer

Search one compound across many targets or scan the strongest compound-target pairs in the active database. The combined reverse-docking score uses a normalized docking-score estimator together with an interaction-fingerprint component.

DB SELECTIONExplorer results are being read from this database.
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2 compounds in matrix 4 best compound-target hits listed 4 targets
• Combined reverse-docking score = 65% normalized docking-score estimator + 35% interaction-fingerprint component.
• When a native ligand exists for an experiment, the interaction-fingerprint component is driven by similarity to the native contact/H-bond pattern.
• When no native ligand exists, the interaction-fingerprint component falls back to contact richness within the experiment (normalized contacts and H-bonds).

Compounds × targets matrix

Each cell shows the best combined reverse-docking score found for that compound on that target. Blank cells mean no imported pose passed the current filters.
Compound Best Mean Targets T03T12T13T20
KB_Leish_190
[H]N(C(=O)[C@@H](C)N([H])c1ccc(C)c(S(=O)(=O)N2CCCCC2)c1)c1ccc(C#N)cc1
0.867 0.856 3 0.85 0.85 0.87
KB_Leish_190
[H]N(C(=O)[C@H](C)N([H])c1ccc(C)c(S(=O)(=O)N2CCCCC2)c1)c1ccc(C#N)cc1
0.852 0.852 1 0.85

Best compound-target hits

The score column is the combined reverse-docking score. The next two columns expose its components: normalized score-estimator and interaction fingerprint.
CompoundTargetExperimentCombinedScore partIFP partIFP modeMetricDock scoreInter normContactsHB
KB_Leish_190
[H]N(C(=O)[C@@H](C)N([H])c1ccc(C)c(S(=O)(=O)N2CCCCC2)c1)c1ccc(C#N)cc1
T20
native IFP available
T20
selection_import_t20
0.867 1.000 0.621 native_similarity final_rank_score -18.2125 -0.644307 12 8 Pose
KB_Leish_190
[H]N(C(=O)[C@@H](C)N([H])c1ccc(C)c(S(=O)(=O)N2CCCCC2)c1)c1ccc(C#N)cc1
T12
native IFP available
T12
selection_import_t12
0.854 1.000 0.584 native_similarity final_rank_score -26.1509 -0.945595 17 8 Pose
KB_Leish_190
[H]N(C(=O)[C@H](C)N([H])c1ccc(C)c(S(=O)(=O)N2CCCCC2)c1)c1ccc(C#N)cc1
T13
native IFP available
T13
selection_import_t13
0.852 1.000 0.577 native_similarity final_rank_score -22.9372 -1.00795 21 8 Pose
KB_Leish_190
[H]N(C(=O)[C@@H](C)N([H])c1ccc(C)c(S(=O)(=O)N2CCCCC2)c1)c1ccc(C#N)cc1
T03
native IFP available
T03
selection_import_t03
0.845 1.000 0.558 native_similarity final_rank_score -23.6416 -0.962761 17 5 Pose