FAIRMol

Reverse docking explorer

Search one compound across many targets or scan the strongest compound-target pairs in the active database. The combined reverse-docking score uses a normalized docking-score estimator together with an interaction-fingerprint component.

DB SELECTIONExplorer results are being read from this database.
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1 compounds in matrix 7 best compound-target hits listed 7 targets
• Combined reverse-docking score = 65% normalized docking-score estimator + 35% interaction-fingerprint component.
• When a native ligand exists for an experiment, the interaction-fingerprint component is driven by similarity to the native contact/H-bond pattern.
• When no native ligand exists, the interaction-fingerprint component falls back to contact richness within the experiment (normalized contacts and H-bonds).

Compounds × targets matrix

Each cell shows the best combined reverse-docking score found for that compound on that target. Blank cells mean no imported pose passed the current filters.
Compound Best Mean Targets T01T02T06T09T10T13T18
KB_HAT_116
[H]O[C@H]1CC[C@H](N([H])c2ncc(Br)c(N([H])c3cccc4c3C(=O)N([H])C4)n2)CC1
0.898 0.840 7 0.84 0.84 0.85 0.77 0.90 0.89 0.79

Best compound-target hits

The score column is the combined reverse-docking score. The next two columns expose its components: normalized score-estimator and interaction fingerprint.
CompoundTargetExperimentCombinedScore partIFP partIFP modeMetricDock scoreInter normContactsHB
KB_HAT_116
[H]O[C@H]1CC[C@H](N([H])c2ncc(Br)c(N([H])c3cccc4c3C(=O)N([H])C4)n2)CC1
T10
native IFP available
T10
selection_import_t10
0.898 1.000 0.708 native_similarity final_rank_score -19.8681 -0.937072 13 12 Pose
KB_HAT_116
[H]O[C@H]1CC[C@H](N([H])c2ncc(Br)c(N([H])c3cccc4c3C(=O)N([H])C4)n2)CC1
T13
native IFP available
T13
selection_import_t13
0.885 1.000 0.672 native_similarity final_rank_score -30.1879 -1.05766 19 9 Pose
KB_HAT_116
[H]O[C@H]1CC[C@H](N([H])c2ncc(Br)c(N([H])c3cccc4c3C(=O)N([H])C4)n2)CC1
T06
native IFP available
T06
selection_import_t06
0.850 1.000 0.570 native_similarity final_rank_score -21.5773 -0.929136 19 1 Pose
KB_HAT_116
[H]O[C@H]1CC[C@H](N([H])c2ncc(Br)c(N([H])c3cccc4c3C(=O)N([H])C4)n2)CC1
T01
native IFP available
T01
selection_import_t01
0.843 1.000 0.552 native_similarity final_rank_score -25.4802 -1.10523 18 7 Pose
KB_HAT_116
[H]O[C@H]1CC[C@H](N([H])c2ncc(Br)c(N([H])c3cccc4c3C(=O)N([H])C4)n2)CC1
T02
native IFP available
T02
selection_import_t02
0.838 1.000 0.539 native_similarity final_rank_score -22.7183 -1.00918 19 7 Pose
KB_HAT_116
[H]O[C@H]1CC[C@H](N([H])c2ncc(Br)c(N([H])c3cccc4c3C(=O)N([H])C4)n2)CC1
T18
native IFP available
T18
selection_import_t18
0.793 1.000 0.408 native_similarity final_rank_score -23.485 -0.88483 14 5 Pose
KB_HAT_116
[H]O[C@H]1CC[C@H](N([H])c2ncc(Br)c(N([H])c3cccc4c3C(=O)N([H])C4)n2)CC1
T09
native IFP available
T09
selection_import_t09
0.772 1.000 0.349 native_similarity final_rank_score -22.4014 -1.01296 18 6 Pose