FAIRMol

Reverse docking explorer

Search one compound across many targets or scan the strongest compound-target pairs in the active database. The combined reverse-docking score uses a normalized docking-score estimator together with an interaction-fingerprint component.

DB SELECTIONExplorer results are being read from this database.
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12 compounds in matrix 54 best compound-target hits listed 19 targets
• Combined reverse-docking score = 65% normalized docking-score estimator + 35% interaction-fingerprint component.
• When a native ligand exists for an experiment, the interaction-fingerprint component is driven by similarity to the native contact/H-bond pattern.
• When no native ligand exists, the interaction-fingerprint component falls back to contact richness within the experiment (normalized contacts and H-bonds).

Compounds × targets matrix

Each cell shows the best combined reverse-docking score found for that compound on that target. Blank cells mean no imported pose passed the current filters.
Compound Best Mean Targets T01T02T03T06T07T08T09T10T11T12T13T14T15T17T18T19T20T21T22
KB_HAT_115 0.952 0.855 7 0.84 0.92 0.95 0.89 0.75 0.73 0.90
KB_HAT_112 0.931 0.850 6 0.83 0.82 0.84 0.79 0.93 0.89
KB_HAT_114 0.922 0.847 6 0.80 0.91 0.84 0.88 0.73 0.92
KB_HAT_110 0.921 0.882 2 0.84 0.92
KB_HAT_114 0.916 0.877 4 0.89 0.92 0.79 0.91
KB_HAT_116 0.898 0.840 7 0.84 0.84 0.85 0.77 0.90 0.89 0.79
KB_HAT_112 0.898 0.838 6 0.85 0.83 0.90 0.80 0.79 0.86
KB_HAT_118 0.887 0.838 7 0.85 0.88 0.82 0.89 0.83 0.81 0.79
KB_HAT_11 0.878 0.845 3 0.85 0.80 0.88
KB_HAT_113 0.858 0.835 4 0.86 0.83 0.82 0.84
KB_HAT_11 0.858 0.858 1 0.86
KB_HAT_119 0.823 0.823 1 0.82

Best compound-target hits

The score column is the combined reverse-docking score. The next two columns expose its components: normalized score-estimator and interaction fingerprint.
CompoundTargetExperimentCombinedScore partIFP partIFP modeMetricDock scoreInter normContactsHB
KB_HAT_115 T10
native IFP available
T10
selection_import_t10
0.952 1.000 0.864 native_similarity final_rank_score -13.2707 -0.942215 17 11 Pose
KB_HAT_112 T21
native IFP available
T21
selection_import_t21
0.931 1.000 0.803 native_similarity final_rank_score -23.1 -0.762765 17 9 Pose
KB_HAT_114 T20
native IFP available
T20
selection_import_t20
0.922 1.000 0.778 native_similarity final_rank_score -22.7724 -0.708568 12 7 Pose
KB_HAT_110 T10
native IFP available
T10
selection_import_t10
0.921 1.000 0.774 native_similarity final_rank_score -21.7069 -0.944906 18 11 Pose
KB_HAT_115 T02
native IFP available
T02
selection_import_t02
0.920 1.000 0.770 native_similarity final_rank_score -23.6644 -1.00152 20 6 Pose
KB_HAT_114 T03
native IFP available
T03
selection_import_t03
0.916 1.000 0.759 native_similarity final_rank_score -26.2166 -0.895312 18 5 Pose
KB_HAT_114 T10
native IFP available
T10
selection_import_t10
0.912 1.000 0.748 native_similarity final_rank_score -30.7847 -0.82574 19 9 Pose
KB_HAT_114 T21
native IFP available
T21
selection_import_t21
0.909 1.000 0.741 native_similarity final_rank_score -25.4939 -0.844229 17 9 Pose
KB_HAT_115 T22
native IFP available
T22
selection_import_t22
0.904 1.000 0.726 native_similarity final_rank_score -24.6608 -1.05438 20 6 Pose
KB_HAT_116 T10
native IFP available
T10
selection_import_t10
0.898 1.000 0.708 native_similarity final_rank_score -19.8681 -0.937072 13 12 Pose
KB_HAT_112 T12
native IFP available
T12
selection_import_t12
0.898 1.000 0.707 native_similarity final_rank_score -23.3712 -0.81121 17 7 Pose
KB_HAT_115 T11
native IFP available
T11
selection_import_t11
0.893 1.000 0.695 native_similarity final_rank_score -19.1155 -0.847649 17 5 Pose
KB_HAT_114 T01
native IFP available
T01
selection_import_t01
0.893 1.000 0.693 native_similarity final_rank_score -23.6981 -0.853403 19 4 Pose
KB_HAT_112 T22
native IFP available
T22
selection_import_t22
0.888 1.000 0.679 native_similarity final_rank_score -32.3861 -1.01947 27 11 Pose
KB_HAT_118 T07
native IFP available
T07
selection_import_t07
0.887 1.000 0.677 native_similarity final_rank_score -35.3362 -1.33485 16 9 Pose
KB_HAT_116 T13
native IFP available
T13
selection_import_t13
0.885 1.000 0.672 native_similarity final_rank_score -30.1879 -1.05766 19 9 Pose
KB_HAT_118 T02
native IFP available
T02
selection_import_t02
0.879 1.000 0.655 native_similarity final_rank_score -22.1541 -1.08501 17 4 Pose
KB_HAT_114 T12
native IFP available
T12
selection_import_t12
0.878 1.000 0.651 native_similarity final_rank_score -21.4609 -0.904408 19 8 Pose
KB_HAT_11 T22
native IFP available
T22
selection_import_t22
0.878 1.000 0.651 native_similarity final_rank_score -27.2061 -1.04405 21 8 Pose
KB_HAT_113 T01
native IFP available
T01
selection_import_t01
0.858 1.000 0.595 native_similarity final_rank_score -21.6122 -1.04464 17 7 Pose
KB_HAT_11 T08
native IFP available
T08
selection_import_t08
0.858 1.000 0.593 native_similarity final_rank_score -33.2334 -1.20877 15 7 Pose
KB_HAT_112 T18
native IFP available
T18
selection_import_t18
0.856 1.000 0.589 native_similarity final_rank_score -19.7275 -0.657056 18 6 Pose
KB_HAT_11 T11
native IFP available
T11
selection_import_t11
0.854 1.000 0.583 native_similarity final_rank_score -21.6675 -0.854516 17 4 Pose
KB_HAT_118 T01
native IFP available
T01
selection_import_t01
0.851 1.000 0.574 native_similarity final_rank_score -25.2784 -1.06423 19 6 Pose
KB_HAT_112 T02
native IFP available
T02
selection_import_t02
0.851 1.000 0.574 native_similarity final_rank_score -27.1849 -0.86795 17 9 Pose
KB_HAT_116 T06
native IFP available
T06
selection_import_t06
0.850 1.000 0.570 native_similarity final_rank_score -21.5773 -0.929136 19 1 Pose
KB_HAT_116 T01
native IFP available
T01
selection_import_t01
0.843 1.000 0.552 native_similarity final_rank_score -25.4802 -1.10523 18 7 Pose
KB_HAT_110 T06
native IFP available
T06
selection_import_t06
0.843 1.000 0.551 native_similarity final_rank_score -20.0202 -0.937167 20 6 Pose
KB_HAT_114 T11
native IFP available
T11
selection_import_t11
0.841 1.000 0.547 native_similarity final_rank_score -33.093 -0.82925 21 3 Pose
KB_HAT_112 T14
native IFP available
T14
selection_import_t14
0.840 1.000 0.542 native_similarity final_rank_score -20.6052 -0.784325 13 8 Pose
KB_HAT_113 T11
native IFP available
T11
selection_import_t11
0.839 1.000 0.539 native_similarity final_rank_score -16.0728 -1.02656 17 6 Pose
KB_HAT_116 T02
native IFP available
T02
selection_import_t02
0.838 1.000 0.539 native_similarity final_rank_score -22.7183 -1.00918 19 7 Pose
KB_HAT_115 T01
native IFP available
T01
selection_import_t01
0.837 1.000 0.535 native_similarity final_rank_score -19.2987 -0.987041 17 7 Pose
KB_HAT_112 T01
native IFP available
T01
selection_import_t01
0.834 1.000 0.526 native_similarity final_rank_score -28.5222 -0.864138 20 5 Pose
KB_HAT_118 T08
native IFP available
T08
selection_import_t08
0.833 1.000 0.523 native_similarity final_rank_score -22.4311 -1.35753 13 12 Pose
KB_HAT_112 T06
native IFP available
T06
selection_import_t06
0.828 1.000 0.510 native_similarity final_rank_score -8.30019 -0.702676 20 2 Pose
KB_HAT_113 T06
native IFP available
T06
selection_import_t06
0.825 1.000 0.500 native_similarity final_rank_score -19.1939 -1.06878 17 5 Pose
KB_HAT_119 T06
native IFP available
T06
selection_import_t06
0.823 1.000 0.495 native_similarity final_rank_score -21.5126 -0.840812 19 3 Pose
KB_HAT_112 T03
native IFP available
T03
selection_import_t03
0.820 1.000 0.486 native_similarity final_rank_score -20.4321 -0.802718 18 3 Pose
KB_HAT_113 T09
native IFP available
T09
selection_import_t09
0.817 1.000 0.478 native_similarity final_rank_score -22.1844 -1.02712 19 7 Pose
KB_HAT_118 T06
native IFP available
T06
selection_import_t06
0.816 1.000 0.475 native_similarity final_rank_score -22.7934 -0.980685 17 4 Pose
KB_HAT_118 T11
native IFP available
T11
selection_import_t11
0.813 1.000 0.465 native_similarity final_rank_score -19.4856 -1.01212 18 4 Pose
KB_HAT_11 T18
native IFP available
T18
selection_import_t18
0.804 1.000 0.441 native_similarity final_rank_score -17.3072 -0.751184 16 3 Pose
KB_HAT_112 T15
native IFP available
T15
selection_import_t15
0.801 1.000 0.431 native_similarity final_rank_score -19.596 -0.737727 17 12 Pose
KB_HAT_114 T02
native IFP available
T02
selection_import_t02
0.798 1.000 0.424 native_similarity final_rank_score -37.2136 -0.931907 18 5 Pose
KB_HAT_112 T17
native IFP available
T17
selection_import_t17
0.793 1.000 0.410 native_similarity final_rank_score -21.541 -0.657785 23 4 Pose
KB_HAT_116 T18
native IFP available
T18
selection_import_t18
0.793 1.000 0.408 native_similarity final_rank_score -23.485 -0.88483 14 5 Pose
KB_HAT_114 T15
native IFP available
T15
selection_import_t15
0.789 1.000 0.397 native_similarity final_rank_score -23.2885 -0.790226 15 5 Pose
KB_HAT_118 T18
native IFP available
T18
selection_import_t18
0.789 1.000 0.397 native_similarity final_rank_score -11.2779 -0.89686 15 5 Pose
KB_HAT_112 T20
native IFP available
T20
selection_import_t20
0.789 1.000 0.396 native_similarity final_rank_score -17.2193 -0.689012 12 9 Pose
KB_HAT_116 T09
native IFP available
T09
selection_import_t09
0.772 1.000 0.349 native_similarity final_rank_score -22.4014 -1.01296 18 6 Pose
KB_HAT_115 T17
native IFP available
T17
selection_import_t17
0.748 1.000 0.279 native_similarity final_rank_score -18.5212 -0.90859 22 8 Pose
KB_HAT_114 T19
native IFP available
T19
selection_import_t19
0.732 1.000 0.234 native_similarity final_rank_score -37.4515 -1.26016 21 7 Pose
KB_HAT_115 T19
native IFP available
T19
selection_import_t19
0.731 1.000 0.232 native_similarity final_rank_score -30.6381 -1.07485 22 7 Pose