FAIRMol

Reverse docking explorer

Search one compound across many targets or scan the strongest compound-target pairs in the active database. The combined reverse-docking score uses a normalized docking-score estimator together with an interaction-fingerprint component.

DB Docking_panel_21Explorer results are being read from this database.
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2 compounds in matrix 9 best compound-target hits listed 9 targets
• Combined reverse-docking score = 65% normalized docking-score estimator + 35% interaction-fingerprint component.
• When a native ligand exists for an experiment, the interaction-fingerprint component is driven by similarity to the native contact/H-bond pattern.
• When no native ligand exists, the interaction-fingerprint component falls back to contact richness within the experiment (normalized contacts and H-bonds).

Compounds × targets matrix

Each cell shows the best combined reverse-docking score found for that compound on that target. Blank cells mean no imported pose passed the current filters.
Compound Best Mean Targets T02T08T13T15T16T18T19T20T21
Z57907181
[H]Oc1cccc([C@H]2c3c(nn([H])c3-c3ccccc3O)C(=O)N2CCc2ccc(OC)c(OC)c2)c1
0.873 0.819 5 0.80 0.85 0.79 0.78 0.87
Z57907181
[H]Oc1cccc([C@@H]2c3c(-c4ccccc4O[H])nn([H])c3C(=O)N2CCc2ccc(OC)c(OC)c2)c1
0.831 0.823 4 0.81 0.83 0.82 0.83

Best compound-target hits

The score column is the combined reverse-docking score. The next two columns expose its components: normalized score-estimator and interaction fingerprint.
CompoundTargetExperimentCombinedScore partIFP partIFP modeMetricDock scoreInter normContactsHB
Z57907181
[H]Oc1cccc([C@H]2c3c(nn([H])c3-c3ccccc3O)C(=O)N2CCc2ccc(OC)c(OC)c2)c1
T21
native IFP available
T21
dockmulti_91311c650f2e_T21
0.873 1.000 0.637 native_similarity final_rank_score -16.9862 -0.668553 17 9 Pose
Z57907181
[H]Oc1cccc([C@H]2c3c(nn([H])c3-c3ccccc3O)C(=O)N2CCc2ccc(OC)c(OC)c2)c1
T15
native IFP available
T15
dockmulti_91311c650f2e_T15
0.852 1.000 0.577 native_similarity final_rank_score -21.9302 -0.571904 15 6 Pose
Z57907181
[H]Oc1cccc([C@@H]2c3c(-c4ccccc4O[H])nn([H])c3C(=O)N2CCc2ccc(OC)c(OC)c2)c1
T20
native IFP available
T20
dockmulti_91311c650f2e_T20
0.831 1.000 0.517 native_similarity final_rank_score -13.5507 -0.437553 10 4 Pose
Z57907181
[H]Oc1cccc([C@@H]2c3c(-c4ccccc4O[H])nn([H])c3C(=O)N2CCc2ccc(OC)c(OC)c2)c1
T13
native IFP available
T13
dockmulti_91311c650f2e_T13
0.826 1.000 0.503 native_similarity final_rank_score -19.5805 -0.710536 19 7 Pose
Z57907181
[H]Oc1cccc([C@@H]2c3c(-c4ccccc4O[H])nn([H])c3C(=O)N2CCc2ccc(OC)c(OC)c2)c1
T18
native IFP available
T18
dockmulti_91311c650f2e_T18
0.824 1.000 0.497 native_similarity final_rank_score -21.9414 -0.613323 12 7 Pose
Z57907181
[H]Oc1cccc([C@@H]2c3c(-c4ccccc4O[H])nn([H])c3C(=O)N2CCc2ccc(OC)c(OC)c2)c1
T08
native IFP available
T08
dockmulti_91311c650f2e_T08
0.811 1.000 0.460 native_similarity final_rank_score -22.8564 -0.800498 13 4 Pose
Z57907181
[H]Oc1cccc([C@H]2c3c(nn([H])c3-c3ccccc3O)C(=O)N2CCc2ccc(OC)c(OC)c2)c1
T02
native IFP available
T02
dockmulti_91311c650f2e_T02
0.802 1.000 0.433 native_similarity final_rank_score -21.3513 -0.741241 17 3 Pose
Z57907181
[H]Oc1cccc([C@H]2c3c(nn([H])c3-c3ccccc3O)C(=O)N2CCc2ccc(OC)c(OC)c2)c1
T16
native IFP available
T16
dockmulti_91311c650f2e_T16
0.786 1.000 0.388 native_similarity final_rank_score -18.5214 -0.500249 13 3 Pose
Z57907181
[H]Oc1cccc([C@H]2c3c(nn([H])c3-c3ccccc3O)C(=O)N2CCc2ccc(OC)c(OC)c2)c1
T19
native IFP available
T19
dockmulti_91311c650f2e_T19
0.783 1.000 0.379 native_similarity final_rank_score -17.6228 -0.686359 13 10 Pose