FAIRMol

Reverse docking explorer

Search one compound across many targets or scan the strongest compound-target pairs in the active database. The combined reverse-docking score uses a normalized docking-score estimator together with an interaction-fingerprint component.

DB Docking_panel_21Explorer results are being read from this database.
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3 compounds in matrix 5 best compound-target hits listed 5 targets
• Combined reverse-docking score = 65% normalized docking-score estimator + 35% interaction-fingerprint component.
• When a native ligand exists for an experiment, the interaction-fingerprint component is driven by similarity to the native contact/H-bond pattern.
• When no native ligand exists, the interaction-fingerprint component falls back to contact richness within the experiment (normalized contacts and H-bonds).

Compounds × targets matrix

Each cell shows the best combined reverse-docking score found for that compound on that target. Blank cells mean no imported pose passed the current filters.
Compound Best Mean Targets T08T09T11T13T19
Z57728363
[H]OCc1cc(=O)c(O[H])c([C@@H](c2cccc(OC)c2)N([H])c2cccc[n+]2[H])o1
0.955 0.925 2 0.96 0.90
Z57728363
[H]OCc1cc(=O)c(O[H])c([C@H](c2cccc(OC)c2)N([H])c2cccc[n+]2[H])o1
0.859 0.828 2 0.86 0.80
Z57728363
[H]OCc1cc(=O)c(O)c([C@H](c2cccc(OC)c2)N([H])c2ccccn2)o1
0.798 0.798 1 0.80

Best compound-target hits

The score column is the combined reverse-docking score. The next two columns expose its components: normalized score-estimator and interaction fingerprint.
CompoundTargetExperimentCombinedScore partIFP partIFP modeMetricDock scoreInter normContactsHB
Z57728363
[H]OCc1cc(=O)c(O[H])c([C@@H](c2cccc(OC)c2)N([H])c2cccc[n+]2[H])o1
T08
native IFP available
T08
dockmulti_91311c650f2e_T08
0.955 1.000 0.873 native_similarity final_rank_score -28.5208 -1.16668 17 7 Pose
Z57728363
[H]OCc1cc(=O)c(O[H])c([C@@H](c2cccc(OC)c2)N([H])c2cccc[n+]2[H])o1
T13
native IFP available
T13
dockmulti_91311c650f2e_T13
0.895 1.000 0.700 native_similarity final_rank_score -20.4441 -0.894227 18 12 Pose
Z57728363
[H]OCc1cc(=O)c(O[H])c([C@H](c2cccc(OC)c2)N([H])c2cccc[n+]2[H])o1
T11
native IFP available
T11
dockmulti_91311c650f2e_T11
0.859 1.000 0.597 native_similarity final_rank_score -20.2699 -0.798467 12 5 Pose
Z57728363
[H]OCc1cc(=O)c(O)c([C@H](c2cccc(OC)c2)N([H])c2ccccn2)o1
T09
native IFP available
T09
dockmulti_91311c650f2e_T09
0.798 1.000 0.424 native_similarity final_rank_score -18.4296 -0.768382 18 4 Pose
Z57728363
[H]OCc1cc(=O)c(O[H])c([C@H](c2cccc(OC)c2)N([H])c2cccc[n+]2[H])o1
T19
native IFP available
T19
dockmulti_91311c650f2e_T19
0.797 1.000 0.419 native_similarity final_rank_score -21.585 -0.860824 12 8 Pose