FAIRMol

Reverse docking explorer

Search one compound across many targets or scan the strongest compound-target pairs in the active database. The combined reverse-docking score uses a normalized docking-score estimator together with an interaction-fingerprint component.

DB Docking_panel_21Explorer results are being read from this database.
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3 compounds in matrix 6 best compound-target hits listed 6 targets
• Combined reverse-docking score = 65% normalized docking-score estimator + 35% interaction-fingerprint component.
• When a native ligand exists for an experiment, the interaction-fingerprint component is driven by similarity to the native contact/H-bond pattern.
• When no native ligand exists, the interaction-fingerprint component falls back to contact richness within the experiment (normalized contacts and H-bonds).

Compounds × targets matrix

Each cell shows the best combined reverse-docking score found for that compound on that target. Blank cells mean no imported pose passed the current filters.
Compound Best Mean Targets T11T14T16T19T20T21
Z56850314
[H]Oc1c([C@@H](c2ccccc2O)N([H])c2nccs2)ccc2cccnc12
0.859 0.824 4 0.86 0.81 0.83 0.79
Z56850314
[H]Oc1ccccc1[C@@H](c1ccc2cccnc2c1O[H])N([H])c1nccs1
0.766 0.766 1 0.77
Z56850314
[H]Oc1ccccc1[C@@H](c1ccc2ccc[n+]([H])c2c1O)N([H])c1nccs1
0.710 0.710 1 0.71

Best compound-target hits

The score column is the combined reverse-docking score. The next two columns expose its components: normalized score-estimator and interaction fingerprint.
CompoundTargetExperimentCombinedScore partIFP partIFP modeMetricDock scoreInter normContactsHB
Z56850314
[H]Oc1c([C@@H](c2ccccc2O)N([H])c2nccs2)ccc2cccnc12
T11
native IFP available
T11
dockmulti_91311c650f2e_T11
0.859 1.000 0.597 native_similarity final_rank_score -21.407 -0.871699 12 5 Pose
Z56850314
[H]Oc1c([C@@H](c2ccccc2O)N([H])c2nccs2)ccc2cccnc12
T20
native IFP available
T20
dockmulti_91311c650f2e_T20
0.834 1.000 0.525 native_similarity final_rank_score -14.4174 -0.69392 6 5 Pose
Z56850314
[H]Oc1c([C@@H](c2ccccc2O)N([H])c2nccs2)ccc2cccnc12
T14
native IFP available
T14
dockmulti_91311c650f2e_T14
0.814 1.000 0.468 native_similarity final_rank_score -17.2871 -0.699454 10 5 Pose
Z56850314
[H]Oc1c([C@@H](c2ccccc2O)N([H])c2nccs2)ccc2cccnc12
T21
native IFP available
T21
dockmulti_91311c650f2e_T21
0.788 1.000 0.394 native_similarity final_rank_score -20.0421 -0.716333 11 5 Pose
Z56850314
[H]Oc1ccccc1[C@@H](c1ccc2cccnc2c1O[H])N([H])c1nccs1
T16
native IFP available
T16
dockmulti_91311c650f2e_T16
0.766 1.000 0.331 native_similarity final_rank_score -20.5643 -0.868428 13 6 Pose
Z56850314
[H]Oc1ccccc1[C@@H](c1ccc2ccc[n+]([H])c2c1O)N([H])c1nccs1
T19
native IFP available
T19
dockmulti_91311c650f2e_T19
0.710 1.000 0.171 native_similarity final_rank_score -35.9316 -1.4015 20 7 Pose