FAIRMol

Reverse docking explorer

Search one compound across many targets or scan the strongest compound-target pairs in the active database. The combined reverse-docking score uses a normalized docking-score estimator together with an interaction-fingerprint component.

DB fairmolExplorer results are being read from this database.
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2 compounds in matrix 7 best compound-target hits listed 7 targets
• Combined reverse-docking score = 65% normalized docking-score estimator + 35% interaction-fingerprint component.
• When a native ligand exists for an experiment, the interaction-fingerprint component is driven by similarity to the native contact/H-bond pattern.
• When no native ligand exists, the interaction-fingerprint component falls back to contact richness within the experiment (normalized contacts and H-bonds).

Compounds × targets matrix

Each cell shows the best combined reverse-docking score found for that compound on that target. Blank cells mean no imported pose passed the current filters.
Compound Best Mean Targets T01T03T09T11T15T17T22
Z56569637
[H]N(/C(O)=C1/C=CC=C/C1=N\S(=O)(=O)c1ccc(F)cc1)c1cc(S(=O)(=O)N2CCCCC2)ccc1Cl
0.887 0.829 4 0.81 0.82 0.79 0.89
Z56569637
[H]N(C(=O)c1ccccc1N([H])S(=O)(=O)c1ccc(F)cc1)c1cc(S(=O)(=O)N2CCCCC2)ccc1Cl
0.873 0.828 3 0.87 0.81 0.80

Best compound-target hits

The score column is the combined reverse-docking score. The next two columns expose its components: normalized score-estimator and interaction fingerprint.
CompoundTargetExperimentCombinedScore partIFP partIFP modeMetricDock scoreInter normContactsHB
Z56569637
[H]N(/C(O)=C1/C=CC=C/C1=N\S(=O)(=O)c1ccc(F)cc1)c1cc(S(=O)(=O)N2CCCCC2)ccc1Cl
T22
native IFP available
T22
selection_import_t22
0.887 1.000 0.678 native_similarity final_rank_score -32.912 -0.852647 21 9 Pose
Z56569637
[H]N(C(=O)c1ccccc1N([H])S(=O)(=O)c1ccc(F)cc1)c1cc(S(=O)(=O)N2CCCCC2)ccc1Cl
T11
native IFP available
T11
selection_import_t11
0.873 1.000 0.637 native_similarity final_rank_score -20.297 -0.664056 12 4 Pose
Z56569637
[H]N(/C(O)=C1/C=CC=C/C1=N\S(=O)(=O)c1ccc(F)cc1)c1cc(S(=O)(=O)N2CCCCC2)ccc1Cl
T03
native IFP available
T03
selection_import_t03
0.823 1.000 0.494 native_similarity final_rank_score -29.0425 -0.931161 19 3 Pose
Z56569637
[H]N(/C(O)=C1/C=CC=C/C1=N\S(=O)(=O)c1ccc(F)cc1)c1cc(S(=O)(=O)N2CCCCC2)ccc1Cl
T01
native IFP available
T01
selection_import_t01
0.812 1.000 0.462 native_similarity final_rank_score -27.092 -0.72614 16 2 Pose
Z56569637
[H]N(C(=O)c1ccccc1N([H])S(=O)(=O)c1ccc(F)cc1)c1cc(S(=O)(=O)N2CCCCC2)ccc1Cl
T15
native IFP available
T15
selection_import_t15
0.809 1.000 0.453 native_similarity final_rank_score -19.7625 -0.708422 15 5 Pose
Z56569637
[H]N(C(=O)c1ccccc1N([H])S(=O)(=O)c1ccc(F)cc1)c1cc(S(=O)(=O)N2CCCCC2)ccc1Cl
T17
native IFP available
T17
selection_import_t17
0.801 1.000 0.432 native_similarity final_rank_score -20.7438 -0.655771 20 5 Pose
Z56569637
[H]N(/C(O)=C1/C=CC=C/C1=N\S(=O)(=O)c1ccc(F)cc1)c1cc(S(=O)(=O)N2CCCCC2)ccc1Cl
T09
native IFP available
T09
selection_import_t09
0.795 1.000 0.413 native_similarity final_rank_score -27.5151 -0.712826 16 2 Pose