FAIRMol

Reverse docking explorer

Search one compound across many targets or scan the strongest compound-target pairs in the active database. The combined reverse-docking score uses a normalized docking-score estimator together with an interaction-fingerprint component.

DB fairmolExplorer results are being read from this database.
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3 compounds in matrix 6 best compound-target hits listed 6 targets
• Combined reverse-docking score = 65% normalized docking-score estimator + 35% interaction-fingerprint component.
• When a native ligand exists for an experiment, the interaction-fingerprint component is driven by similarity to the native contact/H-bond pattern.
• When no native ligand exists, the interaction-fingerprint component falls back to contact richness within the experiment (normalized contacts and H-bonds).

Compounds × targets matrix

Each cell shows the best combined reverse-docking score found for that compound on that target. Blank cells mean no imported pose passed the current filters.
Compound Best Mean Targets T11T14T15T19T20T21
Z56174686
[H]Oc1c([C@H](c2ccccc2F)N([H])c2cc(C)ccn2)ccc2cccnc12
0.902 0.827 4 0.90 0.71 0.80 0.90
Z56174686
[H]Oc1c([C@@H](c2ccccc2F)N([H])c2cc(C)cc[n+]2[H])ccc2cccnc12
0.774 0.774 1 0.77
Z56174686
[H]Oc1c([C@@H](c2ccccc2F)N([H])c2cc(C)ccn2)ccc2cccnc12
0.755 0.755 1 0.76

Best compound-target hits

The score column is the combined reverse-docking score. The next two columns expose its components: normalized score-estimator and interaction fingerprint.
CompoundTargetExperimentCombinedScore partIFP partIFP modeMetricDock scoreInter normContactsHB
Z56174686
[H]Oc1c([C@H](c2ccccc2F)N([H])c2cc(C)ccn2)ccc2cccnc12
T21
native IFP available
T21
selection_import_t21
0.902 1.000 0.719 native_similarity final_rank_score -23.9512 -0.951382 13 7 Pose
Z56174686
[H]Oc1c([C@H](c2ccccc2F)N([H])c2cc(C)ccn2)ccc2cccnc12
T11
native IFP available
T11
selection_import_t11
0.896 1.000 0.702 native_similarity final_rank_score -22.5224 -0.904504 12 7 Pose
Z56174686
[H]Oc1c([C@H](c2ccccc2F)N([H])c2cc(C)ccn2)ccc2cccnc12
T20
native IFP available
T20
selection_import_t20
0.799 1.000 0.425 native_similarity final_rank_score -17.4846 -0.702093 10 6 Pose
Z56174686
[H]Oc1c([C@@H](c2ccccc2F)N([H])c2cc(C)cc[n+]2[H])ccc2cccnc12
T15
native IFP available
T15
selection_import_t15
0.774 1.000 0.353 native_similarity final_rank_score -19.9616 -0.862057 14 3 Pose
Z56174686
[H]Oc1c([C@@H](c2ccccc2F)N([H])c2cc(C)ccn2)ccc2cccnc12
T14
native IFP available
T14
selection_import_t14
0.755 1.000 0.300 native_similarity final_rank_score -23.0264 -0.874055 11 4 Pose
Z56174686
[H]Oc1c([C@H](c2ccccc2F)N([H])c2cc(C)ccn2)ccc2cccnc12
T19
native IFP available
T19
selection_import_t19
0.711 1.000 0.175 native_similarity final_rank_score -30.7727 -1.22901 18 4 Pose