FAIRMol

Reverse docking explorer

Search one compound across many targets or scan the strongest compound-target pairs in the active database. The combined reverse-docking score uses a normalized docking-score estimator together with an interaction-fingerprint component.

DB fairmolExplorer results are being read from this database.
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2 compounds in matrix 16 best compound-target hits listed 16 targets
• Combined reverse-docking score = 65% normalized docking-score estimator + 35% interaction-fingerprint component.
• When a native ligand exists for an experiment, the interaction-fingerprint component is driven by similarity to the native contact/H-bond pattern.
• When no native ligand exists, the interaction-fingerprint component falls back to contact richness within the experiment (normalized contacts and H-bonds).

Compounds × targets matrix

Each cell shows the best combined reverse-docking score found for that compound on that target. Blank cells mean no imported pose passed the current filters.
Compound Best Mean Targets T02T03T05T07T08T10T12T13T15T16T17T18T19T20T21T22
Z49633576
[H]Oc1c(O)ccc(/C=N\Nc2ccc([N+](=O)O)cc2S(=O)(=O)N2CCOCC2)c1O[H]
0.939 0.834 10 0.86 0.75 0.91 0.91 0.94 0.91 0.74 0.79 0.77 0.76
Z49633576
[H]Oc1ccc(/C=[N+](\[H])Nc2ccc([N+](=O)O)cc2S(=O)(=O)N2CCOCC2)c(O[H])c1O[H]
0.928 0.863 6 0.85 0.92 0.77 0.79 0.92 0.93

Best compound-target hits

The score column is the combined reverse-docking score. The next two columns expose its components: normalized score-estimator and interaction fingerprint.
CompoundTargetExperimentCombinedScore partIFP partIFP modeMetricDock scoreInter normContactsHB
Z49633576
[H]Oc1c(O)ccc(/C=N\Nc2ccc([N+](=O)O)cc2S(=O)(=O)N2CCOCC2)c1O[H]
T12
native IFP available
T12
selection_import_t12
0.939 1.000 0.827 native_similarity final_rank_score -23.637 -1.10206 19 16 Pose
Z49633576
[H]Oc1ccc(/C=[N+](\[H])Nc2ccc([N+](=O)O)cc2S(=O)(=O)N2CCOCC2)c(O[H])c1O[H]
T22
native IFP available
T22
selection_import_t22
0.928 1.000 0.794 native_similarity final_rank_score -33.5359 -1.23245 23 14 Pose
Z49633576
[H]Oc1ccc(/C=[N+](\[H])Nc2ccc([N+](=O)O)cc2S(=O)(=O)N2CCOCC2)c(O[H])c1O[H]
T10
native IFP available
T10
selection_import_t10
0.925 1.000 0.785 native_similarity final_rank_score -25.0444 -1.03684 15 11 Pose
Z49633576
[H]Oc1ccc(/C=[N+](\[H])Nc2ccc([N+](=O)O)cc2S(=O)(=O)N2CCOCC2)c(O[H])c1O[H]
T21
native IFP available
T21
selection_import_t21
0.922 1.000 0.776 native_similarity final_rank_score -23.7831 -0.995124 17 11 Pose
Z49633576
[H]Oc1c(O)ccc(/C=N\Nc2ccc([N+](=O)O)cc2S(=O)(=O)N2CCOCC2)c1O[H]
T08
native IFP available
T08
selection_import_t08
0.913 1.000 0.753 native_similarity final_rank_score -35.5119 -1.21638 17 11 Pose
Z49633576
[H]Oc1c(O)ccc(/C=N\Nc2ccc([N+](=O)O)cc2S(=O)(=O)N2CCOCC2)c1O[H]
T13
native IFP available
T13
selection_import_t13
0.908 1.000 0.737 native_similarity final_rank_score -29.3846 -1.04999 17 12 Pose
Z49633576
[H]Oc1c(O)ccc(/C=N\Nc2ccc([N+](=O)O)cc2S(=O)(=O)N2CCOCC2)c1O[H]
T05
native IFP available
T05
selection_import_t05
0.906 1.000 0.732 native_similarity final_rank_score -27.9306 -0.958585 14 8 Pose
Z49633576
[H]Oc1c(O)ccc(/C=N\Nc2ccc([N+](=O)O)cc2S(=O)(=O)N2CCOCC2)c1O[H]
T02
native IFP available
T02
selection_import_t02
0.864 1.000 0.612 native_similarity final_rank_score -17.4184 -0.858251 18 6 Pose
Z49633576
[H]Oc1ccc(/C=[N+](\[H])Nc2ccc([N+](=O)O)cc2S(=O)(=O)N2CCOCC2)c(O[H])c1O[H]
T07
native IFP available
T07
selection_import_t07
0.851 1.000 0.574 native_similarity final_rank_score -26.7529 -1.13727 19 10 Pose
Z49633576
[H]Oc1c(O)ccc(/C=N\Nc2ccc([N+](=O)O)cc2S(=O)(=O)N2CCOCC2)c1O[H]
T17
native IFP available
T17
selection_import_t17
0.791 1.000 0.402 native_similarity final_rank_score -21.8538 -0.756077 17 8 Pose
Z49633576
[H]Oc1ccc(/C=[N+](\[H])Nc2ccc([N+](=O)O)cc2S(=O)(=O)N2CCOCC2)c(O[H])c1O[H]
T20
native IFP available
T20
selection_import_t20
0.786 1.000 0.388 native_similarity final_rank_score -18.0833 -0.734441 7 7 Pose
Z49633576
[H]Oc1c(O)ccc(/C=N\Nc2ccc([N+](=O)O)cc2S(=O)(=O)N2CCOCC2)c1O[H]
T18
native IFP available
T18
selection_import_t18
0.772 1.000 0.348 native_similarity final_rank_score -19.1394 -0.722846 9 4 Pose
Z49633576
[H]Oc1ccc(/C=[N+](\[H])Nc2ccc([N+](=O)O)cc2S(=O)(=O)N2CCOCC2)c(O[H])c1O[H]
T15
native IFP available
T15
selection_import_t15
0.768 1.000 0.337 native_similarity final_rank_score -22.274 -0.832977 10 10 Pose
Z49633576
[H]Oc1c(O)ccc(/C=N\Nc2ccc([N+](=O)O)cc2S(=O)(=O)N2CCOCC2)c1O[H]
T19
native IFP available
T19
selection_import_t19
0.762 1.000 0.319 native_similarity final_rank_score -33.3039 -1.22494 22 11 Pose
Z49633576
[H]Oc1c(O)ccc(/C=N\Nc2ccc([N+](=O)O)cc2S(=O)(=O)N2CCOCC2)c1O[H]
T03
native IFP available
T03
selection_import_t03
0.747 1.000 0.277 native_similarity final_rank_score -22.4387 -1.01606 12 11 Pose
Z49633576
[H]Oc1c(O)ccc(/C=N\Nc2ccc([N+](=O)O)cc2S(=O)(=O)N2CCOCC2)c1O[H]
T16
native IFP available
T16
selection_import_t16
0.743 1.000 0.264 native_similarity final_rank_score -20.3444 -0.914409 15 11 Pose