FAIRMol

Reverse docking explorer

Search one compound across many targets or scan the strongest compound-target pairs in the active database. The combined reverse-docking score uses a normalized docking-score estimator together with an interaction-fingerprint component.

DB Docking_panel_21Explorer results are being read from this database.
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2 compounds in matrix 4 best compound-target hits listed 4 targets
• Combined reverse-docking score = 65% normalized docking-score estimator + 35% interaction-fingerprint component.
• When a native ligand exists for an experiment, the interaction-fingerprint component is driven by similarity to the native contact/H-bond pattern.
• When no native ligand exists, the interaction-fingerprint component falls back to contact richness within the experiment (normalized contacts and H-bonds).

Compounds × targets matrix

Each cell shows the best combined reverse-docking score found for that compound on that target. Blank cells mean no imported pose passed the current filters.
Compound Best Mean Targets T08T12T14T20
Z46080221
[H]N(C(=O)/C(C#N)=C/c1ccc(-c2ccccc2Cl)o1)c1cccc2ncccc12
0.864 0.853 2 0.86 0.84
Z46080221
[H]N(C(=O)/C(C#N)=C\c1ccc(-c2ccccc2Cl)o1)c1cccc2ncccc12
0.830 0.813 2 0.83 0.80

Best compound-target hits

The score column is the combined reverse-docking score. The next two columns expose its components: normalized score-estimator and interaction fingerprint.
CompoundTargetExperimentCombinedScore partIFP partIFP modeMetricDock scoreInter normContactsHB
Z46080221
[H]N(C(=O)/C(C#N)=C/c1ccc(-c2ccccc2Cl)o1)c1cccc2ncccc12
T12
native IFP available
T12
dockmulti_91311c650f2e_T12
0.864 1.000 0.612 native_similarity final_rank_score -23.9977 -0.929235 14 6 Pose
Z46080221
[H]N(C(=O)/C(C#N)=C/c1ccc(-c2ccccc2Cl)o1)c1cccc2ncccc12
T20
native IFP available
T20
dockmulti_91311c650f2e_T20
0.841 1.000 0.546 native_similarity final_rank_score -19.4563 -0.656543 13 4 Pose
Z46080221
[H]N(C(=O)/C(C#N)=C\c1ccc(-c2ccccc2Cl)o1)c1cccc2ncccc12
T08
native IFP available
T08
dockmulti_91311c650f2e_T08
0.830 1.000 0.514 native_similarity final_rank_score -32.1713 -1.07216 14 4 Pose
Z46080221
[H]N(C(=O)/C(C#N)=C\c1ccc(-c2ccccc2Cl)o1)c1cccc2ncccc12
T14
native IFP available
T14
dockmulti_91311c650f2e_T14
0.795 1.000 0.416 native_similarity final_rank_score -23.0122 -0.789348 10 4 Pose