FAIRMol

Reverse docking explorer

Search one compound across many targets or scan the strongest compound-target pairs in the active database. The combined reverse-docking score uses a normalized docking-score estimator together with an interaction-fingerprint component.

DB Docking_panel_21Explorer results are being read from this database.
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2 compounds in matrix 12 best compound-target hits listed 12 targets
• Combined reverse-docking score = 65% normalized docking-score estimator + 35% interaction-fingerprint component.
• When a native ligand exists for an experiment, the interaction-fingerprint component is driven by similarity to the native contact/H-bond pattern.
• When no native ligand exists, the interaction-fingerprint component falls back to contact richness within the experiment (normalized contacts and H-bonds).

Compounds × targets matrix

Each cell shows the best combined reverse-docking score found for that compound on that target. Blank cells mean no imported pose passed the current filters.
Compound Best Mean Targets T02T04T07T08T09T11T12T14T15T18T20T21
Z44848695
[H]Oc1cc(O)ccc1/C=N\N([H])C(=O)c1ccc(CN2C(=O)c3cccc4cccc2c34)cc1
0.945 0.828 8 0.82 0.76 0.85 0.77 0.84 0.87 0.77 0.94
Z44848695
[H]Oc1cc(O)ccc1/C=N/N([H])C(=O)c1ccc(CN2C(=O)c3cccc4cccc2c34)cc1
0.886 0.823 4 0.81 0.84 0.76 0.89

Best compound-target hits

The score column is the combined reverse-docking score. The next two columns expose its components: normalized score-estimator and interaction fingerprint.
CompoundTargetExperimentCombinedScore partIFP partIFP modeMetricDock scoreInter normContactsHB
Z44848695
[H]Oc1cc(O)ccc1/C=N\N([H])C(=O)c1ccc(CN2C(=O)c3cccc4cccc2c34)cc1
T20
native IFP available
T20
dockmulti_91311c650f2e_T20
0.945 1.000 0.842 native_similarity final_rank_score -19.3192 -0.596559 9 4 Pose
Z44848695
[H]Oc1cc(O)ccc1/C=N/N([H])C(=O)c1ccc(CN2C(=O)c3cccc4cccc2c34)cc1
T21
native IFP available
T21
dockmulti_91311c650f2e_T21
0.886 1.000 0.675 native_similarity final_rank_score -27.8344 -0.759998 16 7 Pose
Z44848695
[H]Oc1cc(O)ccc1/C=N\N([H])C(=O)c1ccc(CN2C(=O)c3cccc4cccc2c34)cc1
T12
native IFP available
T12
dockmulti_91311c650f2e_T12
0.866 1.000 0.617 native_similarity final_rank_score -23.9373 -0.687453 16 6 Pose
Z44848695
[H]Oc1cc(O)ccc1/C=N\N([H])C(=O)c1ccc(CN2C(=O)c3cccc4cccc2c34)cc1
T08
native IFP available
T08
dockmulti_91311c650f2e_T08
0.849 1.000 0.568 native_similarity final_rank_score -32.4439 -0.991555 16 5 Pose
Z44848695
[H]Oc1cc(O)ccc1/C=N/N([H])C(=O)c1ccc(CN2C(=O)c3cccc4cccc2c34)cc1
T15
native IFP available
T15
dockmulti_91311c650f2e_T15
0.840 1.000 0.544 native_similarity final_rank_score -17.3649 -0.620321 17 4 Pose
Z44848695
[H]Oc1cc(O)ccc1/C=N\N([H])C(=O)c1ccc(CN2C(=O)c3cccc4cccc2c34)cc1
T11
native IFP available
T11
dockmulti_91311c650f2e_T11
0.835 1.000 0.529 native_similarity final_rank_score -20.841 -0.699602 16 4 Pose
Z44848695
[H]Oc1cc(O)ccc1/C=N\N([H])C(=O)c1ccc(CN2C(=O)c3cccc4cccc2c34)cc1
T02
native IFP available
T02
dockmulti_91311c650f2e_T02
0.822 1.000 0.491 native_similarity final_rank_score -28.9271 -0.921659 15 3 Pose
Z44848695
[H]Oc1cc(O)ccc1/C=N/N([H])C(=O)c1ccc(CN2C(=O)c3cccc4cccc2c34)cc1
T07
native IFP available
T07
dockmulti_91311c650f2e_T07
0.809 1.000 0.453 native_similarity final_rank_score -28.027 -0.938877 15 1 Pose
Z44848695
[H]Oc1cc(O)ccc1/C=N\N([H])C(=O)c1ccc(CN2C(=O)c3cccc4cccc2c34)cc1
T09
native IFP available
T09
dockmulti_91311c650f2e_T09
0.774 1.000 0.353 native_similarity final_rank_score -23.7173 -0.808723 14 3 Pose
Z44848695
[H]Oc1cc(O)ccc1/C=N\N([H])C(=O)c1ccc(CN2C(=O)c3cccc4cccc2c34)cc1
T14
native IFP available
T14
dockmulti_91311c650f2e_T14
0.772 1.000 0.349 native_similarity final_rank_score -22.6903 -0.713098 13 6 Pose
Z44848695
[H]Oc1cc(O)ccc1/C=N\N([H])C(=O)c1ccc(CN2C(=O)c3cccc4cccc2c34)cc1
T04
native IFP available
T04
dockmulti_91311c650f2e_T04
0.762 1.000 0.319 native_similarity final_rank_score -19.1695 -0.553721 13 1 Pose
Z44848695
[H]Oc1cc(O)ccc1/C=N/N([H])C(=O)c1ccc(CN2C(=O)c3cccc4cccc2c34)cc1
T18
native IFP available
T18
dockmulti_91311c650f2e_T18
0.758 1.000 0.309 native_similarity final_rank_score -22.7413 -0.649184 13 2 Pose