FAIRMol

Reverse docking explorer

Search one compound across many targets or scan the strongest compound-target pairs in the active database. The combined reverse-docking score uses a normalized docking-score estimator together with an interaction-fingerprint component.

DB fairmolExplorer results are being read from this database.
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2 compounds in matrix 5 best compound-target hits listed 5 targets
• Combined reverse-docking score = 65% normalized docking-score estimator + 35% interaction-fingerprint component.
• When a native ligand exists for an experiment, the interaction-fingerprint component is driven by similarity to the native contact/H-bond pattern.
• When no native ligand exists, the interaction-fingerprint component falls back to contact richness within the experiment (normalized contacts and H-bonds).

Compounds × targets matrix

Each cell shows the best combined reverse-docking score found for that compound on that target. Blank cells mean no imported pose passed the current filters.
Compound Best Mean Targets T05T08T10T11T14
Z44831560
[H]N(/N=C(\C)c1ccco1)c1cccc(/C(O)=N/N=C(/C)c2ccco2)c1
0.916 0.888 2 0.86 0.92
Z44831560
[H]N(/N=C(\C)c1ccco1)C(=O)c1cccc(N([H])/N=C(/C)c2ccco2)c1
0.914 0.854 3 0.85 0.91 0.80

Best compound-target hits

The score column is the combined reverse-docking score. The next two columns expose its components: normalized score-estimator and interaction fingerprint.
CompoundTargetExperimentCombinedScore partIFP partIFP modeMetricDock scoreInter normContactsHB
Z44831560
[H]N(/N=C(\C)c1ccco1)c1cccc(/C(O)=N/N=C(/C)c2ccco2)c1
T11
native IFP available
T11
selection_import_t11
0.916 1.000 0.761 native_similarity final_rank_score -18.3501 -0.962549 16 3 Pose
Z44831560
[H]N(/N=C(\C)c1ccco1)C(=O)c1cccc(N([H])/N=C(/C)c2ccco2)c1
T10
native IFP available
T10
selection_import_t10
0.914 1.000 0.753 native_similarity final_rank_score -19.5371 -1.00762 17 13 Pose
Z44831560
[H]N(/N=C(\C)c1ccco1)c1cccc(/C(O)=N/N=C(/C)c2ccco2)c1
T08
native IFP available
T08
selection_import_t08
0.859 1.000 0.598 native_similarity final_rank_score -33.6145 -1.2202 14 9 Pose
Z44831560
[H]N(/N=C(\C)c1ccco1)C(=O)c1cccc(N([H])/N=C(/C)c2ccco2)c1
T05
native IFP available
T05
selection_import_t05
0.846 1.000 0.559 native_similarity final_rank_score -27.3019 -1.10642 11 10 Pose
Z44831560
[H]N(/N=C(\C)c1ccco1)C(=O)c1cccc(N([H])/N=C(/C)c2ccco2)c1
T14
native IFP available
T14
selection_import_t14
0.801 1.000 0.432 native_similarity final_rank_score -18.0753 -0.851423 14 7 Pose