FAIRMol

Reverse docking explorer

Search one compound across many targets or scan the strongest compound-target pairs in the active database. The combined reverse-docking score uses a normalized docking-score estimator together with an interaction-fingerprint component.

DB Docking_panel_21Explorer results are being read from this database.
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4 compounds in matrix 4 best compound-target hits listed 4 targets
• Combined reverse-docking score = 65% normalized docking-score estimator + 35% interaction-fingerprint component.
• When a native ligand exists for an experiment, the interaction-fingerprint component is driven by similarity to the native contact/H-bond pattern.
• When no native ligand exists, the interaction-fingerprint component falls back to contact richness within the experiment (normalized contacts and H-bonds).

Compounds × targets matrix

Each cell shows the best combined reverse-docking score found for that compound on that target. Blank cells mean no imported pose passed the current filters.
Compound Best Mean Targets T02T09T16T20
Z31287535
[H]N(/C=C1/C(=O)N(c2ccc(OCC)cc2)C(=O)c2ccccc21)/N=C(\O)[C@@H]1COc2ccccc2O1
0.946 0.946 1 0.95
Z31287535
[H]N(/C=C1\C(=O)N(c2ccc(OCC)cc2)C(=O)c2ccccc21)N([H])C(=O)[C@H]1COc2ccccc2O1
0.901 0.901 1 0.90
Z31287535
[H]N(/C=C1\C(=O)N(c2ccc(OCC)cc2)C(=O)c2ccccc21)/N=C(\O)[C@@H]1COc2ccccc2O1
0.803 0.803 1 0.80
Z31287535
[H]N(/C=C1/C(=O)N(c2ccc(OCC)cc2)C(=O)c2ccccc21)N([H])C(=O)[C@H]1COc2ccccc2O1
0.791 0.791 1 0.79

Best compound-target hits

The score column is the combined reverse-docking score. The next two columns expose its components: normalized score-estimator and interaction fingerprint.
CompoundTargetExperimentCombinedScore partIFP partIFP modeMetricDock scoreInter normContactsHB
Z31287535
[H]N(/C=C1/C(=O)N(c2ccc(OCC)cc2)C(=O)c2ccccc21)/N=C(\O)[C@@H]1COc2ccccc2O1
T20
native IFP available
T20
dockmulti_91311c650f2e_T20
0.946 1.000 0.846 native_similarity final_rank_score -12.145 -0.394438 13 6 Pose
Z31287535
[H]N(/C=C1\C(=O)N(c2ccc(OCC)cc2)C(=O)c2ccccc21)N([H])C(=O)[C@H]1COc2ccccc2O1
T09
native IFP available
T09
dockmulti_91311c650f2e_T09
0.901 1.000 0.717 native_similarity final_rank_score -24.8542 -0.677622 20 4 Pose
Z31287535
[H]N(/C=C1\C(=O)N(c2ccc(OCC)cc2)C(=O)c2ccccc21)/N=C(\O)[C@@H]1COc2ccccc2O1
T16
native IFP available
T16
dockmulti_91311c650f2e_T16
0.803 1.000 0.437 native_similarity final_rank_score -16.4904 -0.553149 14 4 Pose
Z31287535
[H]N(/C=C1/C(=O)N(c2ccc(OCC)cc2)C(=O)c2ccccc21)N([H])C(=O)[C@H]1COc2ccccc2O1
T02
native IFP available
T02
dockmulti_91311c650f2e_T02
0.791 1.000 0.402 native_similarity final_rank_score -19.6393 -0.588478 16 2 Pose